SCHEMBL7658637

SCHEMBL7658637

COc1ccc2c(c1)CC(C(=O)O)N2C(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)C

nearest known ligand 0.58

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CAPN1 P07384 3/20 0.47
CTSL P07711 1/20 0.47
CTSB P07858 1/20 0.47
CTSK P43235 1/20 0.47
CCR1 P32246 2/20 0.47
ACE P12821 2/20 0.46
XIAP P98170 1/20 0.45
CASP1 P29466 1/20 0.44
CASP3 P42574 1/20 0.44
CASP7 P55210 1/20 0.44
CASP6 P55212 1/20 0.44
CASP8 Q14790 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7658633 1.00 CAPN1 (0.47) CAPN1CTSLCTSBCTSKCCR1
SCHEMBL7655796 0.91 ACE (0.51) ACE
SCHEMBL7655799 0.91 ACE (0.51) ACE
SCHEMBL7659034 0.91 ACE (0.51) ACE
SCHEMBL7037763 0.88 KDM4E (0.48) CAPN1CTSLCTSBCTSKCCR1
SCHEMBL3729400 0.88 ACE (0.57) ACEXIAP
SCHEMBL7269341 0.88 ACE (0.57) ACEXIAP
SCHEMBL7039233 0.80 KDM4E (0.50) XIAP
SCHEMBL7043163 0.80 KDM4E (0.50) XIAP
SCHEMBL13260016 0.79 XIAP (0.54) CAPN1CTSLCTSBCTSKCCR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6403561-B1 DISORDERS ASSOCIATED WITH THE INACTIVATION OR EXCESSIVE DEGRADATION OF CHOLECYSTOKININ; INHIBITING THE ENZYMATIC HYDROLYSIS OF CHOLECYSTOKININ 1-(2(S)-AMINOBUTYRYL)-2(S)-INDOLINECARBOXYLIC ACID INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (INSERM) (FR) 2002-06-11 US disclosed