SCHEMBL7659645

SCHEMBL7659645

CCCCNC(=O)N1CCc2ccccc21

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.59
ADRB2 P07550 2/20 0.58
ADRB1 P08588 2/20 0.58
ADRB3 P13945 2/20 0.58
PKM P14618 3/20 0.57
LMNA P02545 1/20 0.56
NPSR1 Q6W5P4 1/20 0.56
NPC1 O15118 3/20 0.56
NFKB1 P19838 3/20 0.56
RAB9A P51151 3/20 0.56
NFKB2 Q00653 3/20 0.56
RELA Q04206 3/20 0.56
SMN1; SMN2 Q16637 3/20 0.56
TP53 P04637 2/20 0.56
NOTUM Q6P988 1/20 0.55
MEN1 O00255 1/20 0.55
KMT2A Q03164 1/20 0.55
POLB P06746 1/20 0.55
TSHR P16473 1/20 0.54
NAMPT P43490 2/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30204966 0.92 MAPT (0.61) MAPTPKMLMNANPSR1NPC1
SCHEMBL14288542 0.86 HSD17B3 (0.58) ADRB2ADRB1ADRB3PKMNAMPT
SCHEMBL4869903 0.86 AVPR2 (0.58) ADRB2ADRB1ADRB3LMNATP53
SCHEMBL4863318 0.86 AVPR2 (0.58) ADRB2ADRB1ADRB3LMNATP53
SCHEMBL157596 0.85 MAPT (0.64) MAPTPKMLMNANPSR1NPC1
SCHEMBL17117468 0.84 MAPT (0.66) MAPTPKMLMNANPSR1NPC1
SCHEMBL7042419 0.83 NOTUM (0.58) MAPTADRB2ADRB1ADRB3NPC1
SCHEMBL17117238 0.83 NPC1 (0.64) MAPTPKMLMNANPSR1NPC1
SCHEMBL4869809 0.82 AVPR2 (0.58) MAPTLMNASMN1; SMN2TP53NOTUM
SCHEMBL1867220 0.81 RAB9A (0.61) MAPTPKMLMNANPSR1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7320993-B1 Aryl-substituted pyridylalkane, alkene, and alkine carboxamides useful as cytostatic useful as cytostatic and immuosuppressive agents ASTELLAS DEUTSCHLAND GMBH (DE) 2008-01-22 US disclosed
US-7320993-B1 Aryl-substituted pyridylalkane, alkene, and alkine carboxamides useful as cytostatic useful as cytostatic and immuosuppressive agents ASTELLAS DEUTSCHLAND GMBH (DE) 2008-01-22 US disclosed
US-6403561-B1 DISORDERS ASSOCIATED WITH THE INACTIVATION OR EXCESSIVE DEGRADATION OF CHOLECYSTOKININ; INHIBITING THE ENZYMATIC HYDROLYSIS OF CHOLECYSTOKININ 1-(2(S)-AMINOBUTYRYL)-2(S)-INDOLINECARBOXYLIC ACID INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (INSERM) (FR) 2002-06-11 US disclosed