SCHEMBL7659783

SCHEMBL7659783

COC(=O)CCc1c(-c2ccc(Cl)cc2)n(C)c2ccncc12

nearest known ligand 0.57

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 17/20 0.57
TBXAS1 P24557 1/20 0.47
CYP11B1 P15538 1/20 0.44
CYP11B2 P19099 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7790361 0.84 TACR1 (0.61) TACR1
SCHEMBL7658708 0.82 TACR1 (0.58) TACR1TBXAS1
SCHEMBL7796987 0.81 TBXAS1 (0.71) TACR1TBXAS1CYP11B1CYP11B2
SCHEMBL7797108 0.80 TACR1 (0.57) TACR1
SCHEMBL7797103 0.80 MAPT (0.54) TACR1
SCHEMBL7797113 0.79 TBXAS1 (0.52) TACR1TBXAS1
SCHEMBL7797019 0.78 TACR1 (0.55) TACR1TBXAS1
SCHEMBL7571685 0.78 TACR1 (0.57) TACR1CYP11B1CYP11B2
SCHEMBL7797005 0.78 TACR1 (0.59) TACR1
SCHEMBL7655822 0.78 TACR1 (0.56) TACR1CYP11B1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6476045-B2 INDOLE AND AZAINDOLE DERIVATIVES AND THEIR USE AS TACHYKININ ANTAGONISTS, AND IN PARTICULAR AS NEUROKININ-1 RECEPTOR ANTAGONIST MERCK SHARP & DOHME LTD. (GB) 2002-11-05 US disclosed