SCHEMBL7662430

SCHEMBL7662430

CC1(C)c2ccccc2NC1C(=O)O

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PDK2 Q15119 1/20 0.40
PDK4 Q16654 1/20 0.40
ALDH1A1 P00352 1/20 0.40
GAA P10253 3/20 0.40
MAPT P10636 1/20 0.40
SMN1; SMN2 Q16637 3/20 0.38
IDO1 P14902 1/20 0.36
TDO2 P48775 1/20 0.36
HSD17B10 Q99714 1/20 0.36
BRD4 O60885 3/20 0.36
CREBBP Q92793 3/20 0.36
EP300 Q09472 1/20 0.36
EGFR P00533 1/20 0.36
KMT2A Q03164 1/20 0.35
BRPF1 P55201 1/20 0.35
CRHBP P24387 1/20 0.35
CRHR2 Q13324 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7662427 1.00 PDK2 (0.40) PDK2PDK4ALDH1A1GAAMAPT
Hydrochloric Acid SCHEMBL10909627 0.98 ALDH1A1 (0.39) PDK2PDK4ALDH1A1GAAMAPT
SCHEMBL9379211 0.84 PDK2 (0.39) PDK2PDK4ALDH1A1GAAMAPT
SCHEMBL10906348 0.84 PDK2 (0.39) PDK2PDK4GAAMAPTSMN1; SMN2
SCHEMBL2001306 0.80 MAPT (0.39) ALDH1A1GAAMAPTSMN1; SMN2IDO1
SCHEMBL18463793 0.79 GAA (0.43) PDK2PDK4ALDH1A1GAAMAPT
SCHEMBL6773255 0.77 KDM4E (0.47) ALDH1A1GAAMAPTSMN1; SMN2IDO1
SCHEMBL16464416 0.77 KDM4E (0.47) ALDH1A1GAAMAPTSMN1; SMN2IDO1
SCHEMBL7043043 0.77 KDM4E (0.47) ALDH1A1GAAMAPTSMN1; SMN2IDO1
SCHEMBL29443040 0.77 KDM4E (0.47) ALDH1A1GAAMAPTSMN1; SMN2IDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6403561-B1 DISORDERS ASSOCIATED WITH THE INACTIVATION OR EXCESSIVE DEGRADATION OF CHOLECYSTOKININ; INHIBITING THE ENZYMATIC HYDROLYSIS OF CHOLECYSTOKININ 1-(2(S)-AMINOBUTYRYL)-2(S)-INDOLINECARBOXYLIC ACID INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (INSERM) (FR) 2002-06-11 US disclosed