SCHEMBL7665402

SCHEMBL7665402

COCCOCCOCCOCCOCCOCCOCCOCCOCCOC(=O)C#Cc1ccc(-c2nc3c(=O)n(CC4CCCCC4)c(=O)n(CC4CCCCC4)c3[nH]2)cc1

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 6/20 0.41
ADORA2B P29275 6/20 0.41
ADORA1 P30542 3/20 0.41
ADORA3 P0DMS8 3/20 0.41
MTOR P42345 8/20 0.34
P2RX3 P56373 3/20 0.33
PIK3CA P42336 2/20 0.31
GSK3A P49840 1/20 0.31
ALDH1A1 P00352 1/20 0.31
PLA2G1B P04054 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
ATG4B Q9Y4P1 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5437774 0.87 ADORA1 (0.43) ADORA2AADORA2BADORA1ADORA3MTOR
SCHEMBL5431586 0.84 ADORA2B (0.53) ADORA2AADORA2BADORA1ADORA3MTOR
SCHEMBL5701832 0.84 ADORA2B (0.53) ADORA2AADORA2BADORA1ADORA3MTOR
SCHEMBL5431701 0.84 ADORA2B (0.53) ADORA2AADORA2BADORA1ADORA3MTOR
SCHEMBL5861429 0.84 ADORA2B (0.53) ADORA2AADORA2BADORA1ADORA3MTOR
SCHEMBL5860233 0.84 ADORA2B (0.53) ADORA2AADORA2BADORA1ADORA3MTOR
SCHEMBL5860446 0.84 ADORA2B (0.53) ADORA2AADORA2BADORA1ADORA3MTOR
SCHEMBL5861492 0.84 ADORA2B (0.53) ADORA2AADORA2BADORA1ADORA3MTOR
SCHEMBL5861525 0.84 ADORA2B (0.53) ADORA2AADORA2BADORA1ADORA3MTOR
SCHEMBL5428341 0.84 ADORA2B (0.53) ADORA2AADORA2BADORA1ADORA3MTOR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6355646-B1 IMMUNOLOGY TREATMENT OF INFLAMMATORY CONDITIONS AND IMMUNE DISORDERS SEPTIC SHOCK GLAXO WELLCOME INC. 2002-03-12 US disclosed