SCHEMBL7669133

SCHEMBL7669133

CCN(CC)CCN(c1ccc2c(c1)nc(CCc1ccc(C(N)=NO)cc1)n2CCC(=O)NC)S(=O)(=O)c1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 4/20 0.43
HDAC8 Q9BY41 3/20 0.43
F2 P00734 7/20 0.42
ALDH1A1 P00352 1/20 0.41
CNR2 P34972 1/20 0.37
THRB P10828 1/20 0.37
RECQL P46063 1/20 0.37
NOS1 P29475 2/20 0.36
OPRM1 P35372 2/20 0.36
NOS3 P29474 1/20 0.36
TXK P42681 1/20 0.36
ITK Q08881 1/20 0.36
GAA P10253 1/20 0.36
BMP1 P13497 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7674611 0.93 HDAC1 (0.43) HDAC1HDAC8F2ALDH1A1THRB
SCHEMBL7664586 0.92 F2 (0.52) HDAC1HDAC8F2ALDH1A1
SCHEMBL7664504 0.90 F2 (0.43) HDAC1HDAC8F2ALDH1A1CNR2
SCHEMBL7664507 0.89 HDAC1 (0.46) HDAC1HDAC8F2ALDH1A1CNR2
SCHEMBL7675369 0.86 F2 (0.41) HDAC1HDAC8F2ALDH1A1CNR2
SCHEMBL7670944 0.85 F2 (0.40) HDAC1HDAC8F2CNR2NOS1
SCHEMBL7672300 0.85 HDAC1 (0.42) HDAC1HDAC8F2ALDH1A1CNR2
SCHEMBL7671039 0.85 F2 (0.53) HDAC1HDAC8F2THRBRECQL
SCHEMBL7667594 0.82 F2 (0.55) HDAC1HDAC8F2CNR2
SCHEMBL7668863 0.82 F2 (0.55) HDAC1HDAC8F2THRBRECQL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6365584-B1 FOR PROPHYLAXIS AND THERAPY OF INFLAMMATORY AND/OR ALLERGIC DISEASES, LUNG FIBROSIS, FIBROSING ALVEOLITIS AND SCARRING, COLLAGENOSES SUCH AS LUPUS ERYTHEMATODES AND SCLERODERMIA AS WELL AS ARTERIOSCLEROSIS, PSORIASIS AND NEOPLASM BOEHRINGER INGELHEIM PHARMA KG (DE) 2002-04-02 US disclosed