SCHEMBL767404

SCHEMBL767404

Fc1nn(C2CCCCO2)c2ccc(Br)cc12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP4F2 P78329 3/20 0.39
CYP4A11 Q02928 3/20 0.39
ALDH1A1 P00352 4/20 0.38
MAPT P10636 3/20 0.38
LMNA P02545 3/20 0.38
MAPK1 P28482 2/20 0.38
TP53 P04637 1/20 0.38
HTT P42858 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
RXRA P19793 1/20 0.36
RXRB P28702 1/20 0.36
RXRG P48443 1/20 0.36
CDK1 P06493 1/20 0.33
RET P07949 2/20 0.33
ALOX15 P16050 1/20 0.32
CNR2 P34972 1/20 0.32
POLB P06746 2/20 0.32
IDO1 P14902 1/20 0.31
EPHX2 P34913 1/20 0.31
ATR Q13535 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15744178 1.00 CYP4F2 (0.39) CYP4F2CYP4A11ALDH1A1MAPTLMNA
SCHEMBL25392984 0.90 CYP4F2 (0.39) CYP4F2CYP4A11ALDH1A1MAPTLMNA
SCHEMBL30182911 0.87 MAPT (0.38) CYP4F2CYP4A11ALDH1A1MAPTLMNA
SCHEMBL18295841 0.85 CYP4F2 (0.39) CYP4F2CYP4A11ALDH1A1MAPTLMNA
SCHEMBL21198696 0.85 CYP4F2 (0.39) CYP4F2CYP4A11ALDH1A1MAPTLMNA
SCHEMBL9904367 0.85 MAPT (0.37) CYP4F2CYP4A11ALDH1A1MAPTLMNA
SCHEMBL24268653 0.85 MAPT (0.37) CYP4F2CYP4A11ALDH1A1MAPTLMNA
SCHEMBL18281904 0.85 GAA (0.41) CYP4F2CYP4A11ALDH1A1MAPTLMNA
SCHEMBL20163477 0.85 CYP4F2 (0.39) CYP4F2CYP4A11ALDH1A1MAPTLMNA
SCHEMBL30615352 0.85 MAPT (0.37) CYP4F2CYP4A11ALDH1A1MAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 80 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12240830-B2 Fused ring heteroaryl compounds and use thereof BISICHEM CO., LTD. (KR) 2025-03-04 US disclosed
EP-4384511-A1 FUSED RING HETEROARYL COMPOUNDS AND USE THEREOF Bisichem Co., Ltd. (KR) 2024-06-19 EP disclosed
EP-4377306-A1 ROCK2 INHIBITORS AND USES THEREOF President and Fellows of Harvard College (US) 2024-06-05 EP disclosed
CN-118055926-A ROCK2 inhibitors and uses thereof 哈佛大学的校长及成员们 2024-05-17 CN disclosed
CN-117881669-A Condensed ring heteroaryl compounds and uses thereof 比西切姆有限公司 2024-04-12 CN disclosed
CN-117529476-A Preparation of substituted 1, 2-diamino heterocyclic derivatives and their use as medicaments 亚飞络思制药公司 2024-02-06 CN disclosed
EP-2735562-B2 Estrogen receptor modulators and uses thereof SERAGON PHARMACEUTICALS INC (US) 2023-11-15 EP disclosed
EP-2735562-B2 Estrogen receptor modulators and uses thereof SERAGON PHARMACEUTICALS INC (US) 2023-11-15 EP disclosed
EP-3544967-B1 SALTS OF INDAZOLE DERIVATIVE AND CRYSTALS THEREOF EISAI R&D MAN CO LTD (JP) 2023-06-28 EP disclosed
US-20230089180-A1 FUSED RING HETEROARYL COMPOUNDS AND USE THEREOF BISICHEM CO., LTD. (KR) 2023-03-23 US disclosed
US-8299112-B2 Estrogen receptor modulators and uses thereof ARAGON PHARMACEUTICALS, INC. (US) 2012-10-30 US disclosed
US-8299112-B2 Estrogen receptor modulators and uses thereof ARAGON PHARMACEUTICALS, INC. (US) 2012-10-30 US disclosed
US-8299112-B2 Estrogen receptor modulators and uses thereof ARAGON PHARMACEUTICALS, INC. (US) 2012-10-30 US disclosed
WO-2012037411-A9 ESTROGEN RECEPTOR MODULATORS AND USES THEREOF ARAGON PHARMACEUTICALS, INC. (US) 2012-05-18 WO disclosed
WO-2012037410-A9 ESTROGEN RECEPTOR MODULATORS AND USES THEREOF ARAGON PHARMACEUTICALS, INC. (US) 2012-05-10 WO disclosed
WO-2012037410-A2 ESTROGEN RECEPTOR MODULATORS AND USES THEREOF ARAGON PHARMACEUTICALS, INC. (US) 2012-03-22 WO disclosed
WO-2012037411-A2 ESTROGEN RECEPTOR MODULATORS AND USES THEREOF ARAGON PHARMACEUTICALS, INC. (US) 2012-03-22 WO disclosed
US-20120071535-A1 ESTROGEN RECEPTOR MODULATORS AND USES THEREOF ARAGON PHARMACEUTICALS, INC. (US) 2012-03-22 US disclosed
US-20120071535-A1 ESTROGEN RECEPTOR MODULATORS AND USES THEREOF ARAGON PHARMACEUTICALS, INC. (US) 2012-03-22 US disclosed
US-20120071535-A1 ESTROGEN RECEPTOR MODULATORS AND USES THEREOF ARAGON PHARMACEUTICALS, INC. (US) 2012-03-22 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230089180-A1 FUSED RING HETEROARYL COMPOUNDS AND USE THEREOF ALK, CYP3A5, SMAD3 CYP4F2 164/4885CYP4A11 42/4885ALDH1A1 727/4885
US-12240830-B2 Fused ring heteroaryl compounds and use thereof ALK, CYP3A5, SMAD3 CYP4F2 164/4885CYP4A11 42/4885ALDH1A1 727/4885
US-20120071535-A1 ESTROGEN RECEPTOR MODULATORS AND USES THEREOF ESR2, ESRRG, GPER1 CYP4F2 604/4885CYP4A11 131/4885ALDH1A1 1178/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.