SCHEMBL7674458

SCHEMBL7674458

O=C(O)c1cc(NS(=O)(=O)c2ccc3ccccc3c2)cc(C(=O)N[C@H](CO)Cc2ccccc2)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 1/20 0.50
PIN1 Q13526 3/20 0.48
SLC16A3 O15427 2/20 0.47
L3MBTL1 Q9Y468 1/20 0.46
F2 P00734 1/20 0.46
ALDH1A1 P00352 2/20 0.46
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
LMNA P02545 1/20 0.46
GAA P10253 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
BACE1 P56817 2/20 0.44
GGPS1 O95749 1/20 0.44
WDR5 P61964 1/20 0.44
GPR27 Q9NS67 1/20 0.43
ROCK2 O75116 1/20 0.43
RPS6KA5 O75582 1/20 0.43
RPS6KA4 O75676 1/20 0.43
PRKACA P17612 1/20 0.43
MAPK1 P28482 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7674462 1.00 AKR1C3 (0.50) AKR1C3PIN1SLC16A3L3MBTL1F2
SCHEMBL7791333 0.89 AKR1C3 (0.54) AKR1C3PIN1SLC16A3F2ALDH1A1
SCHEMBL7791335 0.89 AKR1C3 (0.54) AKR1C3PIN1SLC16A3F2ALDH1A1
SCHEMBL7789327 0.89 ALDH1A1 (0.57) AKR1C3PIN1SLC16A3F2ALDH1A1
SCHEMBL7789330 0.89 ALDH1A1 (0.57) AKR1C3PIN1SLC16A3F2ALDH1A1
SCHEMBL7680207 0.88 AR (0.50) AKR1C3PIN1F2ALDH1A1MEN1
SCHEMBL7680200 0.88 AR (0.50) AKR1C3PIN1F2ALDH1A1MEN1
SCHEMBL7677187 0.85 CAPN1 (0.50) AKR1C3SLC16A3L3MBTL1F2ALDH1A1
SCHEMBL7677185 0.85 CAPN1 (0.50) AKR1C3SLC16A3L3MBTL1F2ALDH1A1
SCHEMBL28666883 0.82 AKR1C3 (0.71) AKR1C3SLC16A3ALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6448254-B1 INHIBITORS OF ENZYMES, IN PARTICULAR CYSTEINE PROTEASES, SUCH AS CALPAIN AND ITS ISOENZYMES AND CATHEPSINS ABBOTT LABORATORIES 2002-09-10 US disclosed