SCHEMBL7674585

SCHEMBL7674585

COc1ccnc(C[O])c1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS2 P35228 11/20 0.62
NOS1 P29475 10/20 0.62
NOS3 P29474 7/20 0.62
CCR1 P32246 1/20 0.55
CCR5 P51681 1/20 0.55
CCR8 P51685 1/20 0.55
CYP2C9 P11712 1/20 0.44
PLAU P00749 1/20 0.43
HTR1A P08908 3/20 0.42
ADRA1D P25100 3/20 0.42
ADRA1A P35348 3/20 0.42
ADRA1B P35368 3/20 0.42
ALDH1A1 P00352 3/20 0.42
MAPT P10636 3/20 0.42
KDM4E B2RXH2 2/20 0.42
CRHBP P24387 1/20 0.42
CRHR2 Q13324 1/20 0.42
HTT P42858 1/20 0.41
PDE8A O60658 1/20 0.41
TP53 P04637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18291870 0.84 NOS2 (0.62) NOS2NOS1NOS3CCR1CCR5
SCHEMBL2760431 0.82 NOS2 (0.65) NOS2NOS1NOS3CCR1CCR5
SCHEMBL29694712 0.80 NOS2 (0.62) NOS2NOS1NOS3CCR1CCR5
SCHEMBL30164187 0.80 NOS2 (0.62) NOS2NOS1NOS3CCR1CCR5
SCHEMBL245100 0.80 NOS2 (0.62) NOS2NOS1NOS3CCR1CCR5
SCHEMBL3307860 0.80 NOS2 (0.62) NOS2NOS1NOS3CCR1CCR5
SCHEMBL1061501 0.80 NOS2 (0.62) NOS2NOS1NOS3CCR1CCR5
SCHEMBL30240847 0.80 NOS2 (0.62) NOS2NOS1NOS3CCR1CCR5
SCHEMBL21847247 0.80 NOS2 (0.62) NOS2NOS1NOS3CCR1CCR5
SCHEMBL11096739 0.80 NOS2 (0.62) NOS2NOS1NOS3CCR1CCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6476021-B1 Compounds having cGMP-PDE inhibitory effect MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 2002-11-05 US disclosed
EP-1048666-A1 NOVEL COMPOUNDS HAVING cGMP-PDE INHIBITORY EFFECT MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 2000-11-02 EP disclosed