SCHEMBL7674732

SCHEMBL7674732

O=C(O)CC1CCC(c2nc(NCc3ccc4c(c3)OCO4)c3c(n2)sc2ccccc23)CC1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.49
PTPN12 Q05209 1/20 0.48
PTPN22 Q9Y2R2 1/20 0.48
SMN1; SMN2 Q16637 2/20 0.47
HTT P42858 3/20 0.46
ALDH1A1 P00352 3/20 0.46
LMNA P02545 1/20 0.46
DGAT1 O75907 1/20 0.45
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
TP53 P04637 1/20 0.44
POLB P06746 1/20 0.44
TSHR P16473 1/20 0.44
MAPK1 P28482 1/20 0.44
HPGD P15428 3/20 0.42
MAPT P10636 2/20 0.42
PDE5A O76074 1/20 0.42
AURKA O14965 1/20 0.41
RPS6KB1 P23443 1/20 0.41
AURKB Q96GD4 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7678118 0.95 GAA (0.44) GAAPTPN12PTPN22SMN1; SMN2HTT
SCHEMBL7674654 0.91 PTPN12 (0.47) GAAPTPN12PTPN22SMN1; SMN2HTT
SCHEMBL6212763 0.90 GAA (0.49) GAAPTPN12PTPN22SMN1; SMN2HTT
Bicarbonate SCHEMBL6214333 0.89 HTT (0.53) GAAPTPN12PTPN22SMN1; SMN2HTT
SCHEMBL7674199 0.87 PDE10A (0.39) GAAPTPN12PTPN22ALDH1A1DGAT1
SCHEMBL6858238 0.87 PDE5A (0.41) ALDH1A1DGAT1PDE5APDE4APDE4B
SCHEMBL6764817 0.86 PTPN12 (0.48) GAAPTPN12PTPN22SMN1; SMN2HTT
SCHEMBL6764845 0.86 PTPN12 (0.45) GAAPTPN12PTPN22SMN1; SMN2HTT
SCHEMBL6852827 0.85 HSD17B10 (0.39) GAAPTPN12PTPN22ALDH1A1DGAT1
SCHEMBL6761170 0.85 GAA (0.43) GAAPTPN12PTPN22SMN1; SMN2HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6495557-B1 SUCH AS 3-(4-(3-CHLORO-4-METHOXYBENZYLAMINO)BENZO-(4,5)-THIENO (2,3-D)PYRIMIDIN-2-YL)PROPIONIC ACID; CARDIOVASCULAR DISORDERS AND/OR IMPAIRED POTENCY MERCK PATENT GESELLSCHAFT MIT BESCHRAENKTER HAFTUNG (DE) 2002-12-17 US disclosed