SCHEMBL6852827

SCHEMBL6852827

O=C(O)CC1CCC(c2nc(NCc3ccc(O)c(Cl)c3)c3c(n2)sc2ccccc23)CC1

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 2/20 0.39
PDE10A Q9Y233 2/20 0.38
STAT6 P42226 2/20 0.36
DGAT1 O75907 5/20 0.36
PDE5A O76074 1/20 0.36
PDE4B Q07343 3/20 0.35
PDE4D Q08499 3/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
HSD17B2 P37059 1/20 0.35
ALDH1A1 P00352 1/20 0.35
GAA P10253 1/20 0.34
PTPN12 Q05209 1/20 0.34
PTPN22 Q9Y2R2 1/20 0.34
EGFR P00533 1/20 0.33
CHRM3 P20309 1/20 0.33
PDE4A P27815 1/20 0.33
PDE4C Q08493 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7674199 0.94 PDE10A (0.39) PDE10ADGAT1PDE5APDE4BPDE4D
SCHEMBL6859354 0.91 HSD17B10 (0.36) HSD17B10PDE10ASTAT6PDE5APDE4B
SCHEMBL6638476 0.90 HSD17B10 (0.40) HSD17B10PDE10ASTAT6PDE5APDE4B
Bicarbonate SCHEMBL6638241 0.89 PDE5A (0.46) HSD17B10PDE10ASTAT6PDE5APDE4B
SCHEMBL6858279 0.89 PDE5A (0.42) PDE5A
SCHEMBL6858238 0.88 PDE5A (0.41) PDE10ADGAT1PDE5APDE4BPDE4D
SCHEMBL6861041 0.88 TRPV1 (0.40)
SCHEMBL7680595 0.88 PDE5A (0.36) PDE10ADGAT1PDE5AALDH1A1
SCHEMBL7403578 0.87 PDE5A (0.46) HSD17B10PDE10ASTAT6PDE5APDE4B
SCHEMBL7675129 0.87 MEN1 (0.39) PDE10ADGAT1PDE5AALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6787548-B1 CARDIOVASCULAR INSUFFICIENCY AND ERECTILE DYSFUNCTION; 3-(4-(3-CHLORO-4-HYDROXYBENZYLAMINO) BENZO(4,5)THIENO(2,3-D)PYRIMIDIN-2-YL)PROPIONIC ACID MERCK Patent Gesellschaft mit beschränkter Haftung (DE) 2004-09-07 US claimed
US-6787548-B1 CARDIOVASCULAR INSUFFICIENCY AND ERECTILE DYSFUNCTION; 3-(4-(3-CHLORO-4-HYDROXYBENZYLAMINO) BENZO(4,5)THIENO(2,3-D)PYRIMIDIN-2-YL)PROPIONIC ACID MERCK Patent Gesellschaft mit beschränkter Haftung (DE) 2004-09-07 US disclosed