SCHEMBL7677331

SCHEMBL7677331

C=CCN(C)CC=CCOc1ccc(C(=O)CC(O)C=C(C)CCC=C(C)C)cc1F

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LSS P48449 5/20 0.40
THRA P10827 1/20 0.35
THRB P10828 1/20 0.35
MTNR1A P48039 1/20 0.35
PTGES O14684 6/20 0.33
KDM4E B2RXH2 1/20 0.32
TRPV1 Q8NER1 1/20 0.32
HDAC3 O15379 1/20 0.31
HDAC4 P56524 1/20 0.31
HDAC1 Q13547 1/20 0.31
HDAC7 Q8WUI4 1/20 0.31
HDAC2 Q92769 1/20 0.31
HDAC10 Q969S8 1/20 0.31
HDAC11 Q96DB2 1/20 0.31
HDAC8 Q9BY41 1/20 0.31
HDAC6 Q9UBN7 1/20 0.31
HDAC9 Q9UKV0 1/20 0.31
HDAC5 Q9UQL6 1/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7677323 1.00 LSS (0.40) LSSTHRATHRBMTNR1APTGES
Fumaric Acid SCHEMBL7681885 0.97 LSS (0.38) LSSTHRATHRBMTNR1APTGES
Fumaric Acid SCHEMBL7681876 0.97 LSS (0.38) LSSTHRATHRBMTNR1APTGES
SCHEMBL7684015 0.90 LSS (0.45) LSSTHRATHRBKDM4EMEN1
SCHEMBL7684020 0.90 LSS (0.45) LSSTHRATHRBKDM4EMEN1
SCHEMBL7769440 0.90 LSS (0.45) LSSTHRATHRBKDM4EMEN1
SCHEMBL7684026 0.90 LSS (0.45) LSSTHRATHRBKDM4EMEN1
Fumaric Acid SCHEMBL7679264 0.87 LSS (0.42) LSSTHRATHRBKDM4EMEN1
Fumaric Acid SCHEMBL7679276 0.87 LSS (0.42) LSSTHRATHRBKDM4EMEN1
SCHEMBL7768105 0.84 PTGES (0.34) THRATHRBMTNR1APTGESKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6441177-B1 Tertiary amines HOFFMANN-LA ROCHE INC. 2002-08-27 US claimed
EP-0778264-B1 Tertiary amines having antimycotic and cholesterol lowering activity HOFFMANN LA ROCHE (CH) 2001-07-11 EP claimed
US-6441177-B1 Tertiary amines HOFFMANN-LA ROCHE INC. 2002-08-27 US disclosed
US-6034275-A FUGICIDES; ATICHOLESTEROL AGENTS HOFFMANN-LA ROCHE INC. (US) 2000-03-07 US disclosed