SCHEMBL7677535

SCHEMBL7677535

NC(=O)c1ccc(-c2ccnc(NCc3ccc(-c4ccc(F)cc4)cc3)n2)cc1.NC(=O)c1ccc(-c2ccnc(NCc3ccc(Br)cc3)n2)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 6/20 0.50
CAMKK2 Q96RR4 5/20 0.50
HDAC3 O15379 3/20 0.50
NCOR1 O75376 3/20 0.50
HDAC2 Q92769 3/20 0.50
GSK3B P49841 2/20 0.50
HDAC8 Q9BY41 2/20 0.50
HDAC6 Q9UBN7 2/20 0.50
MKNK1 Q9BUB5 1/20 0.49
MAPK8 P45983 3/20 0.47
PIK3CG P48736 2/20 0.47
MAPK10 P53779 1/20 0.47
MAPK14 Q16539 1/20 0.45
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
CYP3A4 P08684 1/20 0.44
HDAC11 Q96DB2 1/20 0.44
NCOR2 Q9Y618 1/20 0.44
MAP4K4 O95819 1/20 0.44
CLK1 P49759 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5100599 0.94 CAMKK2 (0.54) HDAC1CAMKK2HDAC3NCOR1HDAC2
SCHEMBL5099819 0.93 HDAC1 (0.56) HDAC1CAMKK2HDAC3NCOR1HDAC2
SCHEMBL5100716 0.84 CAMKK2 (0.50) HDAC1CAMKK2GSK3BMKNK1MAPK8
SCHEMBL5094681 0.83 MAPK8 (0.54) HDAC1CAMKK2HDAC3NCOR1HDAC2
SCHEMBL5091711 0.82 MAPK8 (0.55) HDAC1CAMKK2HDAC3NCOR1HDAC2
SCHEMBL5100280 0.81 HDAC1 (0.53) HDAC1CAMKK2HDAC3NCOR1HDAC2
SCHEMBL5091408 0.81 CAMKK2 (0.54) HDAC1CAMKK2HDAC3NCOR1HDAC2
SCHEMBL5092092 0.79 CLK4 (0.69) HDAC1CAMKK2HDAC3NCOR1HDAC2
SCHEMBL5091615 0.79 HDAC1 (0.54) HDAC1CAMKK2HDAC3NCOR1HDAC2
SCHEMBL5089488 0.79 CAMKK2 (0.61) HDAC1CAMKK2HDAC3NCOR1HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6417185-B1 HETEROCYCLIC ENZYME INHIBITORS CHIRON CORPORATION 2002-07-09 US disclosed