SCHEMBL7677627

SCHEMBL7677627

CN(CC1CC1COc1ccc(C(=O)c2ccc(C#N)cc2)cc1F)C1CC1

nearest known ligand 0.58

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
LSS P48449 8/20 0.58
HRH3 Q9Y5N1 1/20 0.40
NSD2 O96028 3/20 0.38
ACHE P22303 1/20 0.37
VNN1 O95497 1/20 0.35
FASN P49327 1/20 0.35
KDM1A O60341 2/20 0.35
GAA P10253 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
DPP4 P27487 1/20 0.34
DPP9 Q86TI2 1/20 0.34
DPP7 Q9UHL4 1/20 0.34
AR P10275 1/20 0.34
KCNH2 Q12809 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Fumaric Acid SCHEMBL7686380 0.95 LSS (0.53) LSSHRH3NSD2ACHEVNN1
SCHEMBL7683282 0.88 LSS (0.72) LSSACHE
Fumaric Acid SCHEMBL7686204 0.83 LSS (0.65) LSSACHE
SCHEMBL7685852 0.81 LSS (0.57) LSSHRH3NSD2ACHEVNN1
SCHEMBL7685855 0.81 LSS (0.57) LSSHRH3NSD2ACHEVNN1
SCHEMBL7677619 0.80 F10 (0.40) LSSVNN1ARKCNH2
Fumaric Acid SCHEMBL7686378 0.76 F10 (0.37) LSSVNN1AR
SCHEMBL7687794 0.74 LSS (1.00) LSS
SCHEMBL17358775 0.74 LSS (1.00) LSS
Hydrochloric Acid SCHEMBL7687467 0.73 LSS (0.98) LSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6441177-B1 Tertiary amines HOFFMANN-LA ROCHE INC. 2002-08-27 US claimed
EP-0778264-B1 Tertiary amines having antimycotic and cholesterol lowering activity HOFFMANN LA ROCHE (CH) 2001-07-11 EP claimed
US-6441177-B1 Tertiary amines HOFFMANN-LA ROCHE INC. 2002-08-27 US disclosed
US-6034275-A FUGICIDES; ATICHOLESTEROL AGENTS HOFFMANN-LA ROCHE INC. (US) 2000-03-07 US disclosed