SCHEMBL7677619

SCHEMBL7677619

N#Cc1ccc(C(=O)c2ccc(OCC3CC3CNCC3CC3)c(F)c2)cc1

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
F10 P00742 2/20 0.40
VNN1 O95497 5/20 0.39
AR P10275 1/20 0.38
HTR2A P28223 1/20 0.36
LSS P48449 2/20 0.36
SIGMAR1 Q99720 1/20 0.36
PDE4B Q07343 1/20 0.36
USP30 Q70CQ3 1/20 0.35
EGLN2 Q96KS0 1/20 0.35
SCN9A Q15858 1/20 0.35
SLC6A9 P48067 1/20 0.35
KCNH2 Q12809 1/20 0.35
ALDH1A1 P00352 1/20 0.34
MAPT P10636 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Fumaric Acid SCHEMBL7686378 0.94 F10 (0.37) F10VNN1ARHTR2ALSS
SCHEMBL7683275 0.88 LSS (0.45) F10HTR2ALSS
Fumaric Acid SCHEMBL7686200 0.83 LSS (0.42) F10HTR2ALSS
SCHEMBL7685849 0.81 F10 (0.39) F10VNN1ARSIGMAR1USP30
SCHEMBL7677627 0.80 LSS (0.58) VNN1ARLSSKCNH2
Fumaric Acid SCHEMBL7686380 0.76 LSS (0.53) VNN1LSS
SCHEMBL7687793 0.73 LSS (0.61) LSSALDH1A1MAPT
Hydrochloric Acid SCHEMBL7687465 0.72 LSS (0.60) LSSALDH1A1MAPT
SCHEMBL7688273 0.72 LSS (0.67) LSSSCN9AKCNH2
SCHEMBL8047746 0.70 HTT (0.58) VNN1PDE4BALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6441177-B1 Tertiary amines HOFFMANN-LA ROCHE INC. 2002-08-27 US claimed
EP-0778264-B1 Tertiary amines having antimycotic and cholesterol lowering activity HOFFMANN LA ROCHE (CH) 2001-07-11 EP claimed
EP-0778264-A1 Tertiary amines having antimycotic and cholesterol lowering activity F. HOFFMANN-LA ROCHE AG (CH) 1997-06-11 EP claimed
US-6441177-B1 Tertiary amines HOFFMANN-LA ROCHE INC. 2002-08-27 US disclosed
EP-0778264-B1 Tertiary amines having antimycotic and cholesterol lowering activity HOFFMANN LA ROCHE (CH) 2001-07-11 EP disclosed
US-6034275-A FUGICIDES; ATICHOLESTEROL AGENTS HOFFMANN-LA ROCHE INC. (US) 2000-03-07 US disclosed
EP-0778264-A1 Tertiary amines having antimycotic and cholesterol lowering activity F. HOFFMANN-LA ROCHE AG (CH) 1997-06-11 EP disclosed