SCHEMBL7677992

SCHEMBL7677992

CC(Cc1c[nH]c2ccccc12)C(=O)NCc1cccc(Cl)c1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.64
CTDSP1 Q9GZU7 1/20 0.64
MAPT P10636 3/20 0.60
KDM4E B2RXH2 2/20 0.60
MEN1 O00255 1/20 0.60
ALDH1A1 P00352 1/20 0.60
CYP3A4 P08684 1/20 0.60
ALOX15 P16050 1/20 0.60
TSHR P16473 1/20 0.60
MAPK1 P28482 1/20 0.60
KMT2A Q03164 1/20 0.60
HSD17B10 Q99714 1/20 0.60
TDP1 Q9NUW8 1/20 0.60
GABRP O00591 1/20 0.58
GABRD O14764 1/20 0.58
GABRA1 P14867 1/20 0.58
GABRB1 P18505 1/20 0.58
GABRG2 P18507 1/20 0.58
GABRB3 P28472 1/20 0.58
GABRA5 P31644 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7669404 0.88 POLB (0.65) POLBCTDSP1MAPTKDM4EMEN1
SCHEMBL7678136 0.88 POLB (0.67) POLBCTDSP1MAPTKDM4EMEN1
SCHEMBL7838780 0.87 POLB (0.73) POLBCTDSP1MAPTKDM4EMEN1
SCHEMBL7678183 0.87 POLB (0.64) POLBCTDSP1MAPTKDM4EMEN1
SCHEMBL7673231 0.87 POLB (0.64) POLBCTDSP1MAPTKDM4EMEN1
SCHEMBL7677893 0.87 POLB (0.64) POLBCTDSP1MAPTKDM4EMEN1
SCHEMBL7678328 0.86 POLB (0.60) POLBCTDSP1MAPTKDM4EMEN1
SCHEMBL7674758 0.86 MAPT (0.69) POLBCTDSP1MAPTKDM4EMEN1
SCHEMBL7671925 0.85 POLB (0.61) POLBCTDSP1MAPTKDM4EMEN1
SCHEMBL7850770 0.85 POLB (0.61) POLBCTDSP1MAPTKDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6472418-B1 Non-peptide NK1 receptors antagonists WARNER-LAMBERT COMPANY 2002-10-29 US disclosed
EP-1140914-A1 NON-PEPTIDE NK1 RECEPTORS ANTAGONISTS WARNER-LAMBERT COMPANY (US) 2001-10-10 EP disclosed
WO-2000037462-A1 NON-PEPTIDE NK1 RECEPTORS ANTAGONISTS WARNER-LAMBERT COMPANY (US) 2000-06-29 WO disclosed