SCHEMBL7679292

SCHEMBL7679292

c1ccc(CC2CNc3ccc(-c4ccncc4)cc3CN2)cc1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.62
KMT2A Q03164 1/20 0.62
PDE3B Q13370 1/20 0.40
PDE3A Q14432 1/20 0.40
MKNK1 Q9BUB5 1/20 0.36
FNTA P49354 1/20 0.36
FNTB P49356 1/20 0.36
HTR6 P50406 1/20 0.36
IMPDH2 P12268 1/20 0.35
CYP19A1 P11511 1/20 0.35
PRKCI P41743 1/20 0.35
CLK4 Q9HAZ1 3/20 0.34
CHEK1 O14757 2/20 0.34
GSK3B P49841 2/20 0.34
PRKACA P17612 2/20 0.34
CLK2 P49760 2/20 0.34
CDK5 Q00535 2/20 0.34
ROCK1 Q13464 2/20 0.34
DYRK1A Q13627 2/20 0.34
CDK1 P06493 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6633812 1.00 MEN1 (0.62) MEN1KMT2APDE3BPDE3AMKNK1
SCHEMBL6614572 0.92 MEN1 (0.68) MEN1KMT2ACLK4DYRK1BPOLB
SCHEMBL6617044 0.92 MEN1 (0.68) MEN1KMT2ACLK4DYRK1BPOLB
SCHEMBL6617718 0.87 MEN1 (0.55) MEN1KMT2APDE3BPDE3AFNTA
SCHEMBL6614678 0.87 MEN1 (0.58) MEN1KMT2APDE3BPDE3AFNTA
SCHEMBL6616133 0.80 MEN1 (0.68) MEN1KMT2APOLB
SCHEMBL6618053 0.80 MEN1 (0.68) MEN1KMT2APOLB
SCHEMBL6633687 0.80 MEN1 (0.68) MEN1KMT2APOLB
SCHEMBL6615945 0.80 MEN1 (0.68) MEN1KMT2APOLB
SCHEMBL6616489 0.79 MEN1 (0.97) MEN1KMT2APOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6455523-B1 ADMINISTERING 1,4-BENZODIAZEPINE DERIVATIVE AS ANTITUMOR OR ANTICARCINOGENIC AGENT BRISTOL-MYERS SQUIBB COMPANY 2002-09-24 US disclosed
US-6011029-A BENZODIAZEPINE COMPOUNDS BRISTOL-MYERS SQUIBB COMPANY (US) 2000-01-04 US disclosed