SCHEMBL7680075

SCHEMBL7680075

CCCCCc1cn(-c2ccccc2)c(=O)n1Cc1ccc(-c2ncccc2-c2nnn[nH]2)cc1

nearest known ligand 0.51

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
AGTR1 P30556 12/20 0.51
AGTR2 P50052 11/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7686156 0.98 AGTR1 (0.54) AGTR1AGTR2
SCHEMBL7679815 0.94 AGTR1 (0.47) AGTR1AGTR2
SCHEMBL7676512 0.94 AGTR1 (0.51) AGTR1AGTR2
SCHEMBL7684240 0.91 AGTR1 (0.54) AGTR1AGTR2
SCHEMBL9530455 0.90 AGTR1 (0.53) AGTR1AGTR2
SCHEMBL7678948 0.89 AGTR1 (0.49) AGTR1AGTR2
SCHEMBL9555040 0.89 AGTR1 (0.53) AGTR1AGTR2
SCHEMBL7685850 0.88 AGTR1 (0.46) AGTR1AGTR2
SCHEMBL8115702 0.88 AGTR1 (0.55) AGTR1AGTR2
SCHEMBL7681773 0.88 AGTR1 (0.47) AGTR1AGTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6492397-B1 SUCH AS 1-PROPYL-4-BUTYL-1,3-DIHYDRO-3-((5-(2-(1H-TETRAZOL-5-YL)PHENYL)-2 -PYRIDINYL)METHYL)-2H-IMIDAZOL-2-ONE; ANGIO-TENSIN II ANTAGONISTS; CIRCULATORY DISORDERS; HYPERTENSION, CONGESTIVE HEART FAILURE PHARMACIA CORPORATION 2002-12-10 US disclosed
US-5643906-A LOWERING INTRAOCULAR PRESSURE FOR TREATMENT OF GLAUCOMA G.D. SEARLE & CO. (US) 1997-07-01 US disclosed
US-5441970-A Administering angiotensin II antagonists to treat congestive heart failure or hypertension G. D. SEARLE & CO. (US) 1995-08-15 US disclosed
EP-0579766-A1 N-ARYLHETEROARYLALKYL IMIDAZOL-2-ONE COMPOUNDS FOR TREATMENT OF CIRCULATORY DISORDERS G.D. SEARLE & CO. (US) 1994-01-26 EP disclosed
US-5164403-A Hypotensive agents, cardiovascular disorders G. D. SEARLE & CO. (US) 1992-11-17 US disclosed
WO-1992017469-A2 N-ARYLHETEROARYLALKYL IMIDAZOL-2-ONE COMPOUNDS FOR TREATMENT OF CIRCULATORY DISORDERS G.D. SEARLE & CO. (US) 1992-10-15 WO disclosed
EP-0508393-A1 N-arylheteroarylalkyl imidazol-2-one compounds for treatment of circulatory disorders G.D. Searle & Co. (US) 1992-10-14 EP disclosed