SCHEMBL7681554

SCHEMBL7681554

C=CCN(C)CC=CCOc1ccc(C(=O)C=CC=C(C)C)cc1F

nearest known ligand 0.46

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
LSS P48449 12/20 0.46
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
THRA P10827 1/20 0.33
THRB P10828 1/20 0.33
PTPN1 P18031 4/20 0.33
KDM4E B2RXH2 1/20 0.32
LMNA P02545 1/20 0.32
MAPT P10636 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7681546 1.00 LSS (0.46) LSSMEN1KMT2ATHRATHRB
Fumaric Acid SCHEMBL7681356 0.97 LSS (0.44) LSSMEN1KMT2ATHRATHRB
Fumaric Acid SCHEMBL7681358 0.97 LSS (0.44) LSSMEN1KMT2ATHRATHRB
SCHEMBL7681418 0.89 LSS (0.41) LSSTHRATHRBPTPN1LMNA
SCHEMBL7681424 0.89 LSS (0.41) LSSTHRATHRBPTPN1LMNA
Fumaric Acid SCHEMBL7688683 0.87 LSS (0.39) LSSPTPN1
Fumaric Acid SCHEMBL7688682 0.87 LSS (0.39) LSSPTPN1
SCHEMBL7687539 0.85 LSS (0.53) LSSMEN1KMT2ATHRATHRB
SCHEMBL7687535 0.85 LSS (0.53) LSSMEN1KMT2ATHRATHRB
SCHEMBL7688083 0.83 LSS (0.62) LSSPTPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6441177-B1 Tertiary amines HOFFMANN-LA ROCHE INC. 2002-08-27 US claimed
EP-0778264-B1 Tertiary amines having antimycotic and cholesterol lowering activity HOFFMANN LA ROCHE (CH) 2001-07-11 EP claimed
US-6441177-B1 Tertiary amines HOFFMANN-LA ROCHE INC. 2002-08-27 US disclosed
US-6034275-A FUGICIDES; ATICHOLESTEROL AGENTS HOFFMANN-LA ROCHE INC. (US) 2000-03-07 US disclosed