SCHEMBL7681583

SCHEMBL7681583

Cc1ccc(=O)n(CCCN2CCNCC2c2cccc3ccccc23)n1

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 1/20 0.40
TDP1 Q9NUW8 2/20 0.38
HTR2C P28335 8/20 0.35
HTR2A P28223 3/20 0.35
ALDH1A1 P00352 1/20 0.35
ATM Q13315 1/20 0.34
HTR6 P50406 3/20 0.34
HTR2B P41595 2/20 0.34
PKM P14618 1/20 0.34
KCNH2 Q12809 1/20 0.34
IDE P14735 1/20 0.33
UBE2N P61088 1/20 0.33
HTR1A P08908 1/20 0.33
DRD2 P14416 1/20 0.33
HTR1D P28221 1/20 0.33
HTR1B P28222 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7681450 0.98 TAAR1 (0.40) TAAR1TDP1HTR2CHTR2AALDH1A1
SCHEMBL7684227 0.94 TDP1 (0.39) TAAR1TDP1HTR2CHTR2AALDH1A1
SCHEMBL7679337 0.87 CREBBP (0.42) TAAR1PKM
SCHEMBL7681468 0.85 CREBBP (0.42) TAAR1PKM
SCHEMBL7681402 0.81 CREBBP (0.44) ALDH1A1PKM
SCHEMBL8598453 0.80 NPC1 (0.42) TAAR1TDP1HTR2CHTR2AALDH1A1
SCHEMBL8595853 0.78 NPC1 (0.42) TAAR1TDP1HTR2CHTR2AATM
SCHEMBL6164922 0.76 HTR2A (0.45) TAAR1TDP1HTR2CHTR2AHTR2B
SCHEMBL8597121 0.74 NPC1 (0.43) TAAR1TDP1HTR2CHTR2AATM
SCHEMBL8597148 0.73 NPC1 (0.36) TAAR1TDP1HTR2CHTR2AATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6413966-B1 SEROTONERGIC AND CENTRAL DOPAMINERGIC ACTIVITY; AFFINITY FOR 5HT1A AND 5HT2 SEROTONIN AND D2 DOPAMINE RECEPTORS; ATYPICAL ANTIPSYCHOTICS; SCHIZOPHRENIA FAES, FABRICA ESPANOLA DE PRODUCTOS QUIMICOS Y FARMACEUTICOS, S.A. 2002-07-02 US claimed
EP-1057820-A1 Arylpiperazinylalkyl-3(2H)-pyridazinones as serotonin 5HT and dopamine D2 receptor agonists FAES, Fabrica Espanola de Productos Quimicos y Farmaceuticos, S.A. (ES) 2000-12-06 EP claimed