SCHEMBL7681618

SCHEMBL7681618

O=C(O)C1CC1C(=O)NCC1CC1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.47
EPHX1 P07099 2/20 0.46
CYP2C19 P33261 1/20 0.45
GRM4 Q14833 1/20 0.42
CYP2D6 P10635 3/20 0.41
CYP3A4 P08684 3/20 0.41
CYP2C9 P11712 2/20 0.41
TSHR P16473 2/20 0.41
MAPK1 P28482 1/20 0.41
POLB P06746 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.36
ALDH1A1 P00352 1/20 0.36
CA12 O43570 1/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
MMP1 P03956 1/20 0.35
MMP2 P08253 1/20 0.35
MMP3 P08254 1/20 0.35
MMP9 P14780 1/20 0.35
MMP8 P22894 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22277958 0.81 EPHX1 (0.52) TDP1EPHX1CYP2C19GRM4CYP2D6
SCHEMBL22644899 0.79 KDM4E (0.33) TDP1EPHX1CYP2C19GRM4CYP2D6
SCHEMBL13444992 0.78 TDP1 (0.48) TDP1EPHX1CYP2C19GRM4CYP2D6
SCHEMBL13544590 0.75 POLB (0.42) TSHRPOLBTAAR1
SCHEMBL7677400 0.72 POLB (0.51) EPHX1GRM4POLBALDH1A1TAAR1
SCHEMBL3739915 0.72 EPHX1 (0.72) TDP1EPHX1CYP2C19CYP3A4POLB
SCHEMBL4396576 0.71 CYP2D6 (0.63) TDP1EPHX1CYP2C19CYP2D6CYP3A4
SCHEMBL4396572 0.71 CYP2D6 (0.63) TDP1EPHX1CYP2C19CYP2D6CYP3A4
SCHEMBL217411 0.71
SCHEMBL16349314 0.69 GABRR1 (0.53) CYP2C19GRM4CYP2D6CYP2C9TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6441177-B1 Tertiary amines HOFFMANN-LA ROCHE INC. 2002-08-27 US disclosed
US-6034275-A FUGICIDES; ATICHOLESTEROL AGENTS HOFFMANN-LA ROCHE INC. (US) 2000-03-07 US disclosed