SCHEMBL7682184

SCHEMBL7682184

CC(C)(C)c1ccc2[nH]c3c(c2c1)CCNC3C1(C(=O)O)CCC1

nearest known ligand 0.47

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 2/20 0.47
MAPKAPK2 P49137 9/20 0.44
MAPKAPK5 Q8IW41 1/20 0.43
TRPV1 Q8NER1 1/20 0.41
SIRT1 Q96EB6 2/20 0.40
HTR2A P28223 5/20 0.40
HTR2C P28335 4/20 0.40
ALDH1A1 P00352 1/20 0.38
MAPT P10636 1/20 0.38
HTR2B P41595 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7853762 0.90 S1PR1 (0.47) S1PR1MAPKAPK2MAPKAPK5TRPV1SIRT1
SCHEMBL7680950 0.86 SIRT1 (0.54) MAPKAPK2MAPKAPK5SIRT1HTR2AHTR2C
Hydrochloric Acid SCHEMBL7684045 0.86 KMT2A (0.47) S1PR1MAPKAPK2MAPKAPK5TRPV1HTR2A
SCHEMBL7851653 0.85 MAPKAPK2 (0.62) MAPKAPK2SIRT1HTR2AHTR2C
SCHEMBL7843811 0.84 MAPKAPK2 (0.63) MAPKAPK2HTR2AHTR2CHTR2B
SCHEMBL7680354 0.84 HTR2A (0.47) MAPKAPK2MAPKAPK5SIRT1HTR2AHTR2C
SCHEMBL7680308 0.84 MAPKAPK2 (0.63) MAPKAPK2SIRT1HTR2AHTR2CHTR2B
SCHEMBL7681614 0.83 MAPKAPK2 (0.65) MAPKAPK2MAPKAPK5SIRT1HTR2AHTR2C
Hydrochloric Acid SCHEMBL7673540 0.83 HTR2A (0.49) MAPKAPK2MAPKAPK5SIRT1HTR2AHTR2C
Hydrochloric Acid SCHEMBL7673537 0.83 HTR2A (0.49) MAPKAPK2MAPKAPK5SIRT1HTR2AHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6350757-B1 Beta-carboline compounds LES LABORATOIRES SERVIER (FR) 2002-02-26 US disclosed
EP-1070716-A1 Beta-carboline derivatives, process for their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 2001-01-24 EP disclosed