SCHEMBL7682379

SCHEMBL7682379

COC(=O)c1cc(NC(=O)c2ncn(Cc3ccccc3)c2CC2CCCCCC2)cc(C(=O)OC)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.43
LMNA P02545 1/20 0.43
MAPT P10636 1/20 0.43
GAA P10253 1/20 0.41
CASP7 P55210 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
POLB P06746 1/20 0.41
HTT P42858 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
ACKR3 P25106 1/20 0.40
ALDH1A1 P00352 3/20 0.40
PPM1D O15297 1/20 0.40
TP53 P04637 1/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
HSD17B10 Q99714 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
PTPN1 P18031 1/20 0.38
CASR P41180 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6161594 0.91 GAA (0.41) GAAPPM1D
SCHEMBL7682387 0.90 MAPT (0.41) KDM4ELMNAMAPTPOLBALDH1A1
SCHEMBL7083613 0.81 MEN1 (0.41) KDM4EMAPTGAACASP7NPSR1
SCHEMBL7083590 0.78 PKM (0.56) KDM4ELMNAGAANPSR1HTT
SCHEMBL7086563 0.78 CYP19A1 (0.43) LMNAGAAALDH1A1TP53MEN1
SCHEMBL7946943 0.74 CNR1 (0.43) KDM4EMAPTALDH1A1PPM1DSMN1; SMN2
SCHEMBL2367673 0.69 CYP1A2 (0.55) KDM4EMAPTNPSR1POLBHTT
SCHEMBL7688552 0.66 CREBBP (0.43) L3MBTL1
SCHEMBL4150352 0.66 PKM (0.62) GAAALDH1A1SMN1; SMN2IDO1
SCHEMBL4150358 0.65 PKM (0.74) GAAALDH1A1SMN1; SMN2IDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6479531-B1 Gastrin and cholecystokinin receptor ligands JAMES BLACK FOUNDATION LIMITED (GB) 2002-11-12 US disclosed
WO-2001085167-A1 PHARMACEUTICAL COMPOSITIONS COMPRISING PROTON PUMP INHIBITORS AND GASTRIN/CHOLECYSTOKININ RECEPTOR LIGANDS JAMES BLACK FOUNDATION LIMITED (GB) 2001-11-15 WO disclosed