SCHEMBL7683218

SCHEMBL7683218

CCOc1cc(Br)c(N)c(Br)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.46
TDP1 Q9NUW8 1/20 0.46
TP53 P04637 2/20 0.45
CYP3A4 P08684 2/20 0.45
MAPT P10636 5/20 0.44
GAA P10253 2/20 0.44
NQO1 P15559 1/20 0.44
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
NPC1 O15118 1/20 0.41
APOBEC3G Q9HC16 1/20 0.41
CA1 P00915 2/20 0.39
CA2 P00918 2/20 0.39
CA9 Q16790 2/20 0.39
CA12 O43570 1/20 0.39
CA7 P43166 1/20 0.39
NPSR1 Q6W5P4 1/20 0.38
NCOA1 Q15788 1/20 0.38
NCOA3 Q9Y6Q9 1/20 0.38
LMNA P02545 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28191816 0.90 TDP1 (0.42) TSHRTDP1TP53CYP3A4MAPT
SCHEMBL22662565 0.86 CA1 (0.42) TSHRTDP1TP53CYP3A4MAPT
SCHEMBL11399242 0.81 NQO1 (0.48) TSHRTDP1TP53CYP3A4NQO1
SCHEMBL28826529 0.79 NQO1 (0.46) TSHRTDP1TP53CYP3A4MAPT
SCHEMBL26092548 0.78 KDM4E (0.45) TSHRTDP1CYP3A4MAPTGAA
SCHEMBL9172376 0.77 NQO1 (0.44) TSHRTDP1TP53CYP3A4NQO1
SCHEMBL9172372 0.77 NQO1 (0.44) TSHRTDP1TP53CYP3A4MAPT
SCHEMBL4906116 0.77 MEN1 (0.59) TSHRTDP1TP53CYP3A4MAPT
SCHEMBL4889777 0.76 NQO1 (0.42) TSHRTDP1TP53CYP3A4NQO1
SCHEMBL666672 0.75 ALDH1A1 (0.53) TDP1CYP3A4MAPTGAAMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6342503-B1 ANTIDEPRESSANTS, EATING DISORDERS DUPONT PHARMACEUTICALS COMPANY 2002-01-29 US disclosed
US-6107301-A PSYCHOLOGICAL DISORDERS DUPONT PHARMACEUTICALS COMPANY (US) 2000-08-22 US disclosed
EP-0723533-A1 1N-ALKYL-N-ARYLPYRIMIDINAMINES AND DERIVATIVES THEREOF THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1996-07-31 EP disclosed
WO-1995010506-A1 1N-ALKYL-N-ARYLPYRIMIDINAMINES AND DERIVATIVES THEREOF THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1995-04-20 WO disclosed