SCHEMBL7684447

SCHEMBL7684447

CCOc1ccc(-c2ccc3c(c2)C=C(C(=O)Nc2ccc(O)cc2C)CCO3)cc1

nearest known ligand 0.59

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 18/20 0.59
SHMT2 P34897 1/20 0.41
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5204397 0.82 CCR5 (0.72) CCR5NPC1RAB9A
SCHEMBL5205911 0.81 CCR5 (0.71) CCR5NPC1RAB9A
SCHEMBL5551191 0.80 CCR5 (0.55) CCR5NPC1RAB9A
SCHEMBL5205484 0.80 CCR5 (0.56) CCR5NPC1RAB9A
SCHEMBL5210037 0.78 CCR5 (0.56) CCR5
SCHEMBL7685139 0.75 CCR5 (0.53) CCR5
SCHEMBL3034760 0.75 CCR5 (0.73) CCR5
SCHEMBL8122857 0.75 CCR5 (1.00) CCR5
Hydrochloric Acid SCHEMBL3040819 0.74 CCR5 (0.98) CCR5
SCHEMBL7698641 0.74 CCR5 (0.66) CCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6413947-B1 Anilide derivative, production and use thereof TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2002-07-02 US disclosed
EP-1039899-A2 PHARMACEUTICAL COMPOSITION FOR ANTAGONIZING CCR5 COMPRISING ANILIDE DERIVATIVE Takeda Chemical Industries, Ltd. (JP) 2000-10-04 EP disclosed
WO-1999032100-A2 PHARMACEUTICAL COMPOSITION FOR ANTAGONIZING CCR5 COMPRISING ANILIDE DERIVATIVE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1999-07-01 WO disclosed