SCHEMBL7686715

SCHEMBL7686715

CCOC(=O)c1c(-c2ccccc2)nc(C)c(C(=O)O)c1CC

nearest known ligand 0.90

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 16/20 0.90
ALDH1A1 P00352 2/20 0.60
MAPT P10636 2/20 0.60
KDM4E B2RXH2 2/20 0.60
RAB9A P51151 2/20 0.60
LMNA P02545 2/20 0.60
SMN1; SMN2 Q16637 2/20 0.60
NPC1 O15118 1/20 0.60
GAA P10253 1/20 0.60
HPGD P15428 1/20 0.60
NPSR1 Q6W5P4 1/20 0.60
TP53 P04637 1/20 0.54
HSD17B10 Q99714 1/20 0.54
MEN1 O00255 1/20 0.53
KMT2A Q03164 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7678825 0.95 ADORA3 (1.00) ADORA3ALDH1A1MAPTKDM4ERAB9A
SCHEMBL7687342 0.87 ADORA3 (0.83) ADORA3NPSR1
SCHEMBL13780197 0.81 ADORA3 (0.74) ADORA3ALDH1A1MAPTKDM4ERAB9A
SCHEMBL7685833 0.79 ADORA3 (0.76) ADORA3ALDH1A1MAPTKDM4ERAB9A
SCHEMBL30741222 0.78 ADORA3 (1.00) ADORA3NPSR1
SCHEMBL6379843 0.78 ADORA3 (1.00) ADORA3NPSR1
SCHEMBL7681132 0.78 ADORA3 (0.70) ADORA3NPSR1
SCHEMBL7686721 0.78 ADORA3 (1.00) ADORA3ALDH1A1MAPTKDM4ERAB9A
SCHEMBL7682869 0.78 ADORA3 (0.65) ADORA3NPSR1
SCHEMBL7680732 0.77 ADORA3 (1.00) ADORA3NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6376521-B1 ANTIINFLAMMATORY AGENTS; ANTIISCHEMIC AGENTS; CENTRAL NERVOUS SYSTEM DISORDERS THE UNITED STATES OF AMERICA AS REPRESENTED BY THE SECRETARY OF THE DEPARTMENT OF HEALTH AND HUMAN SERVICES 2002-04-23 US disclosed
WO-2000002861-A1 A3 ADENOSINE RECEPTOR ANTAGONISTS THE UNITED STATES OF AMERICA, REPRESENTED BY SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 2000-01-20 WO disclosed