SCHEMBL7687050

SCHEMBL7687050

CCOC(=O)COc1ccc(C(=O)CN2CCN(C3CCN(C(=O)OCCl)CC3)CC2=O)cc1

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.41
HRH3 Q9Y5N1 1/20 0.41
CHRM2 P08172 2/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
GAA P10253 2/20 0.39
ALDH1A1 P00352 4/20 0.39
KDM4E B2RXH2 2/20 0.39
HRH2 P25021 2/20 0.39
HRH1 P35367 2/20 0.39
CHRM1 P11229 1/20 0.39
CHRM3 P20309 1/20 0.39
SMN1; SMN2 Q16637 3/20 0.38
ALOX12 P18054 1/20 0.38
ACHE P22303 2/20 0.38
TSHR P16473 1/20 0.38
MAPT P10636 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7676237 0.90 HRH3 (0.36) CYP2D6HRH3CHRM2L3MBTL1GAA
SCHEMBL7680107 0.90 GAA (0.38) CYP2D6HRH3CHRM2L3MBTL1GAA
SCHEMBL7676228 0.90 CYP2D6 (0.40) CYP2D6HRH3CHRM2L3MBTL1GAA
Hydrochloric Acid SCHEMBL7686863 0.88 CYP2D6 (0.38) CYP2D6HRH3CHRM2L3MBTL1GAA
SCHEMBL7681879 0.88 CYP2D6 (0.38) CYP2D6HRH3CHRM2L3MBTL1GAA
SCHEMBL7676259 0.88 GAA (0.37) CYP2D6HRH3CHRM2L3MBTL1GAA
SCHEMBL7682722 0.88 RAB9A (0.36) CYP2D6HRH3ALDH1A1KDM4EHRH2
Hydrochloric Acid SCHEMBL7684461 0.87 CYP2D6 (0.38) CYP2D6HRH3CHRM2L3MBTL1GAA
SCHEMBL7687250 0.87 GAA (0.36) CYP2D6HRH3CHRM2GAAALDH1A1
SCHEMBL7686845 0.87 HRH2 (0.38) CYP2D6HRH3CHRM2L3MBTL1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6472397-B1 Nitrogen-containing heterocyclic compounds having antiplatelet aggregation effect and medicinal use thereof MEIJI SEIKA KAISHA, LTD. (JP) 2002-10-29 US disclosed
EP-1070712-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUNDS HAVING ANTIPLATELET AGGREGATION EFFECT AND MEDICINAL USE THEREOF MEIJI SEIKA KAISHA LTD. (JP) 2001-01-24 EP disclosed