SCHEMBL76877

SCHEMBL76877

COC(=O)CN(C(=O)[C@H]1C[C@@H](OCC(C)(C)C)CN1C(=O)O)c1ccc(N2CCOCC2=O)cc1

nearest known ligand 0.45

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
F10 P00742 19/20 0.45
MLYCD O95822 1/20 0.36
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3103779 0.90 F10 (0.46) F10MLYCDCYP1A2CYP3A4CYP2D6
SCHEMBL76876 0.84 F10 (0.46) F10MLYCDCYP1A2CYP3A4CYP2D6
SCHEMBL77721 0.81 F10 (0.66) F10
SCHEMBL85545 0.78 F10 (0.64) F10
SCHEMBL4214502 0.78 F10 (0.43) F10MLYCDCYP1A2CYP3A4CYP2D6
SCHEMBL76878 0.73 F10 (0.38) F10MLYCDCYP1A2CYP3A4CYP2D6
SCHEMBL3096939 0.70 F10 (0.65) F10
SCHEMBL3114123 0.66 F10 (0.61) F10
SCHEMBL7734355 0.66 F10 (0.45) F10CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL78227 0.66 F10 (0.84) F10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8129373-B2 Carbonyl compounds MERCK PATENT GMBH (DE) 2012-03-06 US disclosed