SCHEMBL7689896

SCHEMBL7689896

CCCCC(NC(=O)c1ccccc1C=Cc1ccc(CN(C)C)cc1)C(=O)CNC(C)=O

nearest known ligand 0.75

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CAPN1 P07384 13/20 0.75
CTSB P07858 7/20 0.75
CTSS P25774 2/20 0.49
CTSK P43235 2/20 0.49
CTSL P07711 2/20 0.44
HDAC3 O15379 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
MMP13 P45452 1/20 0.36
EHMT2 Q96KQ7 3/20 0.36
MMP2 P08253 1/20 0.33
MMP3 P08254 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7693912 0.91 CAPN1 (0.73) CAPN1CTSBCTSSCTSKCTSL
SCHEMBL7696167 0.89 CAPN1 (0.57) CAPN1CTSBCTSSCTSKCTSL
SCHEMBL7698259 0.87 CAPN1 (0.61) CAPN1CTSBCTSSCTSKCTSL
SCHEMBL7696527 0.86 CAPN1 (0.65) CAPN1CTSBCTSSCTSKCTSL
SCHEMBL7695427 0.85 CAPN1 (0.56) CAPN1CTSBCTSSCTSKCTSL
SCHEMBL7692161 0.85 CAPN1 (0.70) CAPN1CTSBCTSSCTSKCTSL
SCHEMBL7691158 0.84 CAPN1 (0.54) CAPN1CTSBCTSSCTSKCTSL
SCHEMBL7696093 0.84 CAPN1 (0.54) CAPN1CTSBCTSSCTSKCTSL
SCHEMBL1930492 0.84 CAPN1 (0.86) CAPN1CTSBCTSSCTSKCTSL
SCHEMBL1930489 0.84 CAPN1 (0.86) CAPN1CTSBCTSSCTSKCTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6436925-B1 BETTER ABLE TO CROSS MEMBRANES; INHIBITORS OF CYSTEINE PROTEASES LIKE CALPAIN I AND II AND CATHEPSIN B AND L, CAN THUS BE USED TO CONTROL DISEASES ASSOCIATED WITH AN ELEVATED ACTIVITY OF CALPAIN ENZYMES OR CATHEPSIN ENZYMES ABBOTT LABORATORIES 2002-08-20 US disclosed