SCHEMBL7698259

SCHEMBL7698259

CC(=O)NCC(=O)[C@H](Cc1ccccc1)NC(=O)c1ccccc1C=Cc1ccc(CN(C)C)cc1

nearest known ligand 0.61

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CAPN1 P07384 13/20 0.61
CTSB P07858 7/20 0.61
CTSS P25774 2/20 0.60
CTSK P43235 2/20 0.60
CTSL P07711 2/20 0.54
ITGB1 P05556 1/20 0.41
ITGA4 P13612 1/20 0.41
ITGB7 P26010 1/20 0.41
PTPN1 P18031 2/20 0.39
MMP13 P45452 1/20 0.39
RAB9A P51151 1/20 0.38
HDAC3 O15379 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7696964 0.92 CAPN1 (0.61) CAPN1CTSBCTSSCTSKCTSL
SCHEMBL7688883 0.91 CAPN1 (0.75) CAPN1CTSBCTSSCTSKCTSL
SCHEMBL7690823 0.90 CAPN1 (0.60) CAPN1CTSBCTSSCTSKCTSL
SCHEMBL7689896 0.87 CAPN1 (0.75) CAPN1CTSBCTSSCTSKCTSL
SCHEMBL7694140 0.87 CAPN1 (0.60) CAPN1CTSBCTSSCTSKCTSL
SCHEMBL7688501 0.86 CAPN1 (0.58) CAPN1CTSBCTSSCTSKCTSL
SCHEMBL7697556 0.86 CAPN1 (0.53) CAPN1CTSBCTSSCTSKCTSL
SCHEMBL7697899 0.85 CAPN1 (0.53) CAPN1CTSBCTSSCTSKCTSL
SCHEMBL7697767 0.84 CAPN1 (0.54) CAPN1CTSBCTSSCTSKCTSL
SCHEMBL7695603 0.84 CAPN1 (0.70) CAPN1CTSBCTSSCTSKCTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6436925-B1 BETTER ABLE TO CROSS MEMBRANES; INHIBITORS OF CYSTEINE PROTEASES LIKE CALPAIN I AND II AND CATHEPSIN B AND L, CAN THUS BE USED TO CONTROL DISEASES ASSOCIATED WITH AN ELEVATED ACTIVITY OF CALPAIN ENZYMES OR CATHEPSIN ENZYMES ABBOTT LABORATORIES 2002-08-20 US disclosed