SCHEMBL7694334

SCHEMBL7694334

CC(=O)NCC(=O)[C@H](Cc1ccccc1)NC(=O)c1cccc(NS(=O)(=O)c2ccccc2)c1

nearest known ligand 0.50

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.49
CTSD P07339 1/20 0.49
BACE1 P56817 1/20 0.49
BACE2 Q9Y5Z0 1/20 0.49
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
KDM1A O60341 2/20 0.47
MAOA P21397 1/20 0.47
PTGES O14684 1/20 0.46
PFKFB3 Q16875 1/20 0.46
EGFR P00533 1/20 0.46
FGFR1 P11362 1/20 0.46
KDR P35968 1/20 0.46
HDAC2 Q92769 1/20 0.45
HDAC8 Q9BY41 1/20 0.45
HDAC6 Q9UBN7 1/20 0.45
ACE P12821 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7695659 0.92 KDM1A (0.51) ALDH1A1CTSDBACE1BACE2MEN1
SCHEMBL7695396 0.91 AKR1C3 (0.48) ALDH1A1MEN1KMT2AHDAC2HDAC8
SCHEMBL7665441 0.87 EGFR (0.46) MEN1KMT2AKDM1AMAOAPFKFB3
SCHEMBL7689353 0.86 ALDH1A1 (0.44) ALDH1A1MEN1KMT2APFKFB3
SCHEMBL7692550 0.82 AKR1C3 (0.51) ALDH1A1CTSDBACE1BACE2MEN1
SCHEMBL7689558 0.81 ALDH1A1 (0.55) ALDH1A1MEN1KMT2AHDAC2HDAC8
SCHEMBL7694179 0.80 AKR1C3 (0.48) ALDH1A1
SCHEMBL7661487 0.80 EGFR (0.47) MEN1KMT2AKDM1AMAOAPTGES
SCHEMBL7696803 0.78 ALDH1A1 (0.44) ALDH1A1MEN1KMT2AKDM1AMAOA
SCHEMBL7378076 0.77 CAPN1 (0.53) CTSDBACE1BACE2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6436925-B1 BETTER ABLE TO CROSS MEMBRANES; INHIBITORS OF CYSTEINE PROTEASES LIKE CALPAIN I AND II AND CATHEPSIN B AND L, CAN THUS BE USED TO CONTROL DISEASES ASSOCIATED WITH AN ELEVATED ACTIVITY OF CALPAIN ENZYMES OR CATHEPSIN ENZYMES ABBOTT LABORATORIES 2002-08-20 US disclosed