SCHEMBL7696233

SCHEMBL7696233

CC(CNc1ccc(-c2n[nH]c3c2Cc2ccccc2-3)cc1)N1CCN(C)CC1

nearest known ligand 0.62

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KDR P35968 13/20 0.62
CHEK1 O14757 5/20 0.51
CDK1 P06493 1/20 0.50
CDK2 P24941 1/20 0.50
KCNH2 Q12809 1/20 0.44
KIT P10721 1/20 0.41
FLT1 P17948 1/20 0.41
FLT4 P35916 1/20 0.41
TEK Q02763 1/20 0.41
PDGFRB P09619 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7704710 0.92 KDR (0.54) KDRCHEK1CDK1CDK2PDGFRB
SCHEMBL7701433 0.91 KDR (0.53) KDRCHEK1CDK1CDK2KCNH2
SCHEMBL7704425 0.90 KDR (0.52) KDRCHEK1CDK1CDK2
SCHEMBL7701582 0.84 KDR (0.70) KDRCHEK1CDK1CDK2KCNH2
SCHEMBL7701118 0.78 KDR (0.61) KDRCHEK1CDK1CDK2KIT
SCHEMBL7090562 0.77 KDR (0.60) KDRCHEK1CDK1CDK2
SCHEMBL6999873 0.77 KDR (0.50) KDRCHEK1CDK1CDK2KCNH2
SCHEMBL7000955 0.77 KDR (0.65) KDRCHEK1CDK1CDK2KIT
SCHEMBL7090565 0.76 KDR (0.59) KDRCHEK1CDK1CDK2KCNH2
SCHEMBL7091164 0.75 CHEK1 (0.50) KDRCHEK1CDK1CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6462036-B1 INHIBITING SIGNAL TRANSDUCTION BY MODULATING ACTIVITY OF RECEPTOR AND NONRECEPTOR TYROSINE AND SERINE/THREONINE KINASES TO REGULATE AND MODULATE ABNORMAL OR INAPPROPRIATE CELL PROLIFERATION, DIFFERENTIATION, OR METABOLISM BASF AKTIENGESELLSCHAFT (DE) 2002-10-08 US disclosed