SCHEMBL7696937

SCHEMBL7696937

O=C(Nc1ccccc1OC[C@H](O)CN1CCC(n2c(=O)[nH]c3cc(C(F)(F)F)ccc32)CC1)c1ccccc1

nearest known ligand 0.52

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
OPRL1 P41146 2/20 0.52
PLD2 O14939 8/20 0.49
PLD1 Q13393 7/20 0.49
SCN1A P35498 5/20 0.49
SCN5A Q14524 5/20 0.49
SCN9A Q15858 5/20 0.49
HSD11B1 P28845 2/20 0.46
TNKS O95271 1/20 0.45
PARP1 P09874 1/20 0.45
PARP2 Q9UGN5 1/20 0.45
CALCRL Q16602 1/20 0.44
CTSS P25774 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4804251 1.00 OPRL1 (0.52) OPRL1PLD2PLD1SCN1ASCN5A
SCHEMBL4803925 0.94 PLD2 (0.55) OPRL1PLD2PLD1
SCHEMBL4806688 0.92 OPRL1 (0.54) OPRL1PLD2PLD1SCN1ASCN5A
SCHEMBL4805216 0.92 PLD2 (0.59) OPRL1PLD2PLD1SCN1ASCN5A
Hydrochloric Acid SCHEMBL4806574 0.89 OPRL1 (0.61) OPRL1PLD2PLD1SCN1ASCN5A
SCHEMBL4807512 0.86 PLD2 (0.66) OPRL1PLD2PLD1
SCHEMBL4804373 0.86 PLD2 (0.60) OPRL1PLD2PLD1HSD11B1
SCHEMBL4806305 0.85 PLD2 (0.59) OPRL1PLD2PLD1HSD11B1
SCHEMBL4806019 0.83 OPRL1 (0.63) OPRL1PLD2PLD1CTSS
SCHEMBL4807271 0.83 OPRL1 (0.67) OPRL1PLD2PLD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002074763-A9 BENZIMIDAZOL DERIVATIVES MODULATE CHEMOKINE RECEPTORS ASTRAZENECA AB (SE) 2002-10-24 WO disclosed