SCHEMBL7698643

SCHEMBL7698643

COc1ccc(N2C(=O)c3cc(CN4Cc5cnc(N)cc5C4=O)ccc3C2C)cc1OC(C)CCc1ccccc1

nearest known ligand 0.35

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 1/20 0.35
NR1H3 Q13133 1/20 0.35
TNIK Q9UKE5 3/20 0.34
PDE4A P27815 3/20 0.34
PDE4B Q07343 3/20 0.34
PDE4C Q08493 3/20 0.34
PDE4D Q08499 3/20 0.34
MCHR1 Q99705 1/20 0.34
EGFR P00533 8/20 0.33
ROCK2 O75116 1/20 0.33
ROCK1 Q13464 1/20 0.33
HTR2C P28335 1/20 0.33
HTR2B P41595 1/20 0.33
CACNA2D1 P54289 1/20 0.32
TRPC6 Q9Y210 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7700346 0.92 NR1H2 (0.35) NR1H2NR1H3TNIKPDE4APDE4B
SCHEMBL7693775 0.89 MCHR1 (0.44) NR1H2NR1H3PDE4APDE4BPDE4C
SCHEMBL7703112 0.89 NR1H2 (0.38) NR1H2NR1H3PDE4APDE4BPDE4C
SCHEMBL7699521 0.87 PDE4A (0.35) NR1H2NR1H3PDE4APDE4BPDE4C
SCHEMBL7698759 0.86 PDE4A (0.38) NR1H2NR1H3PDE4APDE4BPDE4C
SCHEMBL7698210 0.84 PDE4B (0.43) PDE4APDE4BPDE4CPDE4DHTR2C
SCHEMBL7700309 0.81 MCHR1 (0.44) NR1H2NR1H3PDE4APDE4BPDE4C
SCHEMBL7699082 0.81 MCHR1 (0.43) NR1H2NR1H3PDE4APDE4BPDE4C
SCHEMBL7694958 0.81 NR1H3 (0.44) NR1H2NR1H3PDE4APDE4BPDE4C
SCHEMBL7700767 0.80 MCHR1 (0.42) NR1H2NR1H3PDE4APDE4BPDE4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002081446-A1 3-CYCLOPENTYLOXY-4-METHOXYPHENYL-ISOINDOLINONE DERIVATIVES AND THE USE THEREOF DAEWOONG CO., LTD. (KR) 2002-10-17 WO disclosed