SCHEMBL7700494

SCHEMBL7700494

NC(=O)c1cccc2nc(N3CCN(CCc4ccc([N+](=O)[O-])cc4)CC3)[nH]c12

nearest known ligand 0.51

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
KCNJ1 P48048 17/20 0.51
KCNH2 Q12809 16/20 0.51
SIGMAR1 Q99720 1/20 0.47
HRH3 Q9Y5N1 1/20 0.46
CYP3A4 P08684 1/20 0.43
ABCC1 P33527 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7700401 0.96 HRH3 (0.48) KCNJ1KCNH2SIGMAR1HRH3CYP3A4
SCHEMBL7700409 0.87 CYP3A4 (0.44) CYP3A4ABCC1
SCHEMBL7706360 0.86 CYP3A4 (0.43) HRH3CYP3A4ABCC1
SCHEMBL7708429 0.86 CYP3A4 (0.43) CYP3A4ABCC1
SCHEMBL7700403 0.86 CYP3A4 (0.43) CYP3A4ABCC1
SCHEMBL7700417 0.86 CYP2C9 (0.48) SIGMAR1CYP3A4ABCC1
SCHEMBL7700415 0.86 CYP3A4 (0.45) SIGMAR1CYP3A4ABCC1
SCHEMBL5621658 0.86 PARP1 (0.56) KCNJ1KCNH2
SCHEMBL7702657 0.84 PARP1 (0.42) KCNH2CYP3A4ABCC1
SCHEMBL7708443 0.84 KCNH2 (0.48) KCNJ1KCNH2SIGMAR1CYP3A4ABCC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6448271-B1 SUCH AS 2-(PIPERIDIN-4-YL)BENZIMIDAZOLE-4-CARBOXAMIDE; INHIBITORS OF ENZYME POLY(ADP-RIBOSE)POLYMERASE; IMPROVED WATER SOLUBILITY BASF AKTIENGESELLSCHAFT (DE) 2002-09-10 US disclosed