SCHEMBL7708443

SCHEMBL7708443

N#Cc1ccc(CCN2CCN(c3nc4cccc(C(N)=O)c4[nH]3)CC2)cc1

nearest known ligand 0.48

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 8/20 0.48
KCNJ1 P48048 5/20 0.48
PARP1 P09874 7/20 0.48
ADRA1D P25100 1/20 0.43
ADRA1A P35348 1/20 0.43
ADRA1B P35368 1/20 0.43
CYP3A4 P08684 1/20 0.42
ABCC1 P33527 1/20 0.42
DRD4 P21917 1/20 0.41
SLC6A2 P23975 1/20 0.41
HTR1D P28221 1/20 0.41
HTR2A P28223 1/20 0.41
HTR2C P28335 1/20 0.41
SLC6A4 P31645 1/20 0.41
HTR7 P34969 1/20 0.41
HTR2B P41595 1/20 0.41
TMEM97 Q5BJF2 1/20 0.41
SIGMAR1 Q99720 1/20 0.41
PARP2 Q9UGN5 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7705645 0.96 PARP1 (0.45) KCNH2KCNJ1PARP1ADRA1DADRA1A
SCHEMBL7700409 0.88 CYP3A4 (0.44) PARP1CYP3A4ABCC1SLC6A4
SCHEMBL7700417 0.87 CYP2C9 (0.48) PARP1CYP3A4ABCC1DRD4SLC6A2
SCHEMBL7700415 0.87 CYP3A4 (0.45) PARP1ADRA1DADRA1AADRA1BCYP3A4
SCHEMBL7706360 0.87 CYP3A4 (0.43) PARP1ADRA1DADRA1AADRA1BCYP3A4
SCHEMBL7700403 0.87 CYP3A4 (0.43) PARP1ADRA1DADRA1AADRA1BCYP3A4
SCHEMBL7708429 0.87 CYP3A4 (0.43) PARP1CYP3A4ABCC1HTR2AHTR2C
SCHEMBL5621936 0.86 PARP1 (0.65) PARP1
SCHEMBL7702682 0.85 SIGMAR1 (0.48) KCNH2KCNJ1PARP1ADRA1DADRA1A
SCHEMBL5621724 0.85 CYP3A4 (0.44) PARP1ADRA1DADRA1AADRA1BCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6448271-B1 SUCH AS 2-(PIPERIDIN-4-YL)BENZIMIDAZOLE-4-CARBOXAMIDE; INHIBITORS OF ENZYME POLY(ADP-RIBOSE)POLYMERASE; IMPROVED WATER SOLUBILITY BASF AKTIENGESELLSCHAFT (DE) 2002-09-10 US disclosed