SCHEMBL7701225

SCHEMBL7701225

CCOCC1(C)CCCSc2cc(C#Cc3ccc(C(=O)OC(=O)c4ccc(C#Cc5ccc6c(c5)SCCCC6(C)COC)cc4)cc3)ccc21

nearest known ligand 0.41

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
RARB P10826 13/20 0.41
RARG P13631 13/20 0.41
RARA P10276 10/20 0.41
CYP3A4 P08684 4/20 0.41
KMT2A Q03164 1/20 0.41
CYP26A1 O43174 2/20 0.35
CRABP2 P29373 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7701222 0.92 RARB (0.45) RARBRARGRARACYP3A4KMT2A
SCHEMBL7140735 0.89 RARB (0.40) RARBRARGRARACYP3A4KMT2A
SCHEMBL7142149 0.88 RARB (0.48) RARBRARGRARACYP3A4KMT2A
SCHEMBL7136046 0.86 RARB (0.50) RARBRARGRARACYP3A4KMT2A
SCHEMBL7143911 0.77 RARB (0.45) RARBRARGRARACYP3A4KMT2A
SCHEMBL7143918 0.77 RARB (0.45) RARBRARGRARACYP3A4KMT2A
SCHEMBL9007003 0.73 RARB (0.66) RARBRARGRARACYP3A4KMT2A
SCHEMBL7136227 0.72 RARA (0.48) RARBRARGRARACYP3A4CYP26A1
SCHEMBL7139166 0.72 RARA (0.48) RARBRARGRARACYP3A4CYP26A1
SCHEMBL7139242 0.71

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1212316-A2 BENZOPYRANS AND BENZOTHIOPYRANS AS RAR SELECTIVE RETINOID AGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2002-06-12 EP claimed
WO-2001014360-A2 BENZOPYRANS AND BENZOTHIOPYRANS AS RAR SELECTIVE RETINOID AGONISTS F. HOFFMAN-LA ROCHE AG (CH) 2001-03-01 WO claimed