SCHEMBL7701573

SCHEMBL7701573

FC(F)(F)c1cccc(N2CCN(Cc3nc4ccccc4n3CN3C=CON3)CC2)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM2 Q14416 6/20 0.48
DRD4 P21917 4/20 0.48
ALDH1A2 O94788 1/20 0.47
ALDH1A1 P00352 1/20 0.47
ALDH2 P05091 1/20 0.47
ALDH3A1 P30838 1/20 0.47
ALDH1A3 P47895 1/20 0.47
DRD2 P14416 2/20 0.45
TP53 P04637 2/20 0.44
KDM4E B2RXH2 3/20 0.44
OPRM1 P35372 2/20 0.44
OPRD1 P41143 1/20 0.44
DRD3 P35462 2/20 0.44
MAPT P10636 2/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
ABCB11 O95342 1/20 0.44
HTR1A P08908 1/20 0.44
ADRA2A P08913 1/20 0.44
ADORA3 P0DMS8 1/20 0.44
CHRM1 P11229 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6095533 0.78 DRD4 (0.56) GRM2DRD4ALDH1A2ALDH1A1ALDH2
SCHEMBL6095488 0.77 GRM2 (0.50) GRM2DRD4ALDH1A2ALDH1A1ALDH2
SCHEMBL15748175 0.71 SIGMAR1 (0.58) DRD2OPRM1DRD3ABCB11HTR1A
SCHEMBL15748232 0.69 SIGMAR1 (0.59) DRD2OPRM1DRD3ABCB11HTR1A
SCHEMBL17471515 0.69 DRD3 (0.56) GRM2DRD4ALDH1A1DRD2TP53
SCHEMBL6095407 0.67 DRD4 (0.64) GRM2DRD4DRD2MAPTSMN1; SMN2
Hydrochloric Acid SCHEMBL7695313 0.67 KDM4E (0.57) ALDH1A1DRD2TP53KDM4EDRD3
SCHEMBL11925196 0.67 DRD3 (0.54) GRM2DRD4ALDH1A1DRD2TP53
SCHEMBL6864697 0.67 SIGMAR1 (0.76) DRD4ALDH1A1DRD2TP53KDM4E
SCHEMBL7859184 0.66 PHGDH (0.58) GRM2DRD4ALDH1A1DRD2TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002092575-A1 BENZIMIDAZOLE COMPOUNDS AND ANTIVIRAL USES THEREOF TRIMERIS, INC. (US) 2002-11-21 WO disclosed