SCHEMBL7701983

SCHEMBL7701983

CC(C)Oc1ccc[c]c1-c1ccccc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IRAK4 Q9NWZ3 2/20 0.42
ALDH1A1 P00352 3/20 0.37
ACHE P22303 1/20 0.37
S1PR1 P21453 1/20 0.36
S1PR3 Q99500 1/20 0.36
HTR1A P08908 1/20 0.36
TLR8 Q9NR97 1/20 0.36
MCHR1 Q99705 1/20 0.36
HDAC4 P56524 1/20 0.35
KDM4E B2RXH2 2/20 0.35
LMNA P02545 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
HPGD P15428 1/20 0.34
GAA P10253 1/20 0.33
ADRA2A P08913 1/20 0.33
ADRA2B P18089 1/20 0.33
ADRA2C P18825 1/20 0.33
NISCH Q9Y2I1 1/20 0.33
ADRA1D P25100 1/20 0.33
ADRA1A P35348 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1274782 0.79 CA1 (0.46) ALDH1A1KDM4ELMNATDP1HPGD
SCHEMBL7459866 0.79 IDO1 (0.36) ALDH1A1TDP1HPGDADRA2BCYP1A2
SCHEMBL2091154 0.76 TSHR (0.42) ALDH1A1HTR1ALMNAHPGDGAA
SCHEMBL11382454 0.75 ALDH1A1 (0.44) ALDH1A1HTR1AKDM4ETDP1ADRA1D
SCHEMBL7006398 0.75 CA1 (0.38) IRAK4ALDH1A1ACHEKDM4ETDP1
SCHEMBL1819088 0.73 IRAK4 (0.39) IRAK4ALDH1A1ACHEHTR1ATLR8
SCHEMBL16960318 0.73 IRAK4 (0.39) IRAK4ALDH1A1ACHEHTR1ATLR8
SCHEMBL161636 0.72 IRAK4 (0.38) IRAK4ALDH1A1ACHETLR8MCHR1
SCHEMBL16962525 0.72 IRAK4 (0.38) IRAK4ALDH1A1ACHEHTR1ATLR8
SCHEMBL9673377 0.72 IRAK4 (0.42) IRAK4ALDH1A1ACHEHTR1ATLR8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1242399-A1 $g(a)-ARYLETHYLPIPERAZINE DERIVATIVES AS NEUROKININ ANTAGONISTS UCB S.A. (BE) 2002-09-25 EP disclosed
WO-2001046167-A1 α-ARYLETHYLPIPERAZINE DERIVATIVES AS NEUROKININ ANTAGONISTS UCB, S.A. (BE) 2001-06-28 WO disclosed