SCHEMBL7702013

SCHEMBL7702013

NC(=O)CN1CCN(C(Cc2ccc(C(N)=O)cc2)OCc2cc(C(F)(F)F)cc(C(F)(F)F)c2)CC1

nearest known ligand 0.55

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 18/20 0.55
MAOB P27338 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7705814 0.82 TACR1 (0.52) TACR1
SCHEMBL6480881 0.80 TACR1 (0.82) TACR1
SCHEMBL7705392 0.74 TACR1 (0.52) TACR1MAOB
SCHEMBL6481341 0.73 TACR1 (0.80) TACR1
SCHEMBL6488715 0.71 TACR1 (1.00) TACR1
SCHEMBL6488713 0.71 TACR1 (1.00) TACR1
SCHEMBL7705623 0.67 TACR1 (0.56) TACR1
SCHEMBL2780550 0.66 DDR1 (0.54) TACR1
SCHEMBL6861962 0.65 KDM4E (0.63) TACR1
Water SCHEMBL6479022 0.64 TACR1 (0.82) TACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1242399-A1 $g(a)-ARYLETHYLPIPERAZINE DERIVATIVES AS NEUROKININ ANTAGONISTS UCB S.A. (BE) 2002-09-25 EP disclosed
WO-2001046167-A1 α-ARYLETHYLPIPERAZINE DERIVATIVES AS NEUROKININ ANTAGONISTS UCB, S.A. (BE) 2001-06-28 WO disclosed