SCHEMBL6861962

SCHEMBL6861962

NC(=O)CN1CCN(Cc2cccc(C(F)(F)F)c2)CC1

nearest known ligand 0.63

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.63
ALDH1A1 P00352 2/20 0.63
GAA P10253 2/20 0.63
ATM Q13315 1/20 0.62
LMNA P02545 2/20 0.61
FAAH O00519 2/20 0.60
SIGMAR1 Q99720 2/20 0.56
PARP1 P09874 1/20 0.54
DRD4 P21917 2/20 0.53
KMT2A Q03164 2/20 0.52
ACHE P22303 1/20 0.52
HTT P42858 1/20 0.52
MEN1 O00255 1/20 0.51
TACR1 P25103 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30747663 0.86 FAAH (0.67) KDM4EALDH1A1GAAATMLMNA
SCHEMBL16217376 0.86 MEN1 (0.48) KDM4EALDH1A1GAAATMLMNA
SCHEMBL6865563 0.84 FAAH (0.61) KDM4EALDH1A1GAALMNAFAAH
SCHEMBL2929974 0.82 FAAH (0.72) KDM4EALDH1A1GAALMNAFAAH
SCHEMBL6865538 0.82 ALDH1A1 (0.47) KDM4EALDH1A1LMNAKMT2AHTT
SCHEMBL21297283 0.82 ALDH1A1 (0.47) KDM4EALDH1A1KMT2AHTTMEN1
SCHEMBL31414613 0.82 SIGMAR1 (0.63) KDM4EALDH1A1GAAATMLMNA
SCHEMBL1761024 0.81 FAAH (0.67) KDM4EALDH1A1GAALMNAFAAH
SCHEMBL6865561 0.80 FAAH (0.59) KDM4EALDH1A1GAALMNAFAAH
SCHEMBL4244138 0.79 ALDH1A1 (0.97) KDM4EALDH1A1GAALMNAFAAH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5817489-A BACTERICIDES, OR CHEMICAL INTERMEDIATES THEREOF; DRUG LIBRARIES ISIS PHARMACEUTICALS, INC. (US) 1998-10-06 US claimed
US-6800444-B1 USEFUL AS ANTIBACTERIAL AND OTHER PHARMACEUTICAL AGENTS/INTERMEDIATES ISIS PHARMACEUTICALS, INC. 2004-10-05 US disclosed
US-6660466-B1 Reacting reactive appendage compounds such as meta benzylic compounds or alpha-amide compounds with scaffold molecules having reactive functionalities and contacting the intermediate library with a reducing agent ISIS PHARMACEUTICALS, INC. 2003-12-09 US disclosed
US-5922872-A BACTERICIDES AND DRUGS ISIS PHARMACEUTICALS, INC. (US) 1999-07-13 US disclosed
US-5817489-A BACTERICIDES, OR CHEMICAL INTERMEDIATES THEREOF; DRUG LIBRARIES ISIS PHARMACEUTICALS, INC. (US) 1998-10-06 US disclosed
US-5798360-A ANTIBACTERIAL AGENTS ISIS PHARMACEUTICALS, INC. (US) 1998-08-25 US disclosed
US-5780241-A ALTERING ELECTROCHEMICAL PROPERTIES BY DECYCLIZATION ISIS PHARMACEUTICALS, INC. (US) 1998-07-14 US disclosed
WO-1998020349-A1 COMPLEX CHEMICAL LIBRARIES ISIS PHARMACEUTICALS, INC. (US) 1998-05-14 WO disclosed
US-5731438-A BACTERICIDES; DRUGS ISIS PHARMACEUTICALS, INC. (US) 1998-03-24 US disclosed
WO-1998005332-A1 NOVEL HETEROCYCLE COMPOSITIONS ISIS PHARMACEUTICALS, INC. (US) 1998-02-12 WO disclosed