SCHEMBL7702982

SCHEMBL7702982

N=C(N)NC(=O)C1=Cc2cccc(C(=O)NC(=N)N)c2OCC1

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 3/20 0.43
NPC1 O15118 2/20 0.34
RAB9A P51151 2/20 0.34
KMT2A Q03164 1/20 0.34
SSTR4 P31391 3/20 0.32
TP53 P04637 1/20 0.32
MAPT P10636 2/20 0.32
POLB P06746 1/20 0.32
HTT P42858 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
NPSR1 Q6W5P4 1/20 0.30
RXFP1 Q9HBX9 1/20 0.30
PTGES O14684 1/20 0.30
CA12 O43570 1/20 0.30
CA9 Q16790 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7697554 0.99 PARP1 (0.42) PARP1NPC1RAB9AKMT2ASSTR4
SCHEMBL7701178 0.93 PARP1 (0.41) PARP1NPC1RAB9AKMT2ATP53
SCHEMBL7697131 0.89 PARP1 (0.46) PARP1NPC1RAB9AKMT2ATP53
SCHEMBL7702986 0.89 PARP1 (0.38) PARP1NPC1RAB9AKMT2ASSTR4
Hydrochloric Acid SCHEMBL7702260 0.88 PARP1 (0.36) PARP1NPC1KMT2ATP53HTT
SCHEMBL7700738 0.88 PARP1 (0.37) PARP1NPC1RAB9AKMT2ATP53
Hydrochloric Acid SCHEMBL7697560 0.88 PARP1 (0.37) PARP1NPC1RAB9AKMT2ASSTR4
SCHEMBL7694851 0.87 PARP1 (0.36) PARP1NPC1RAB9AKMT2ATP53
Hydrochloric Acid SCHEMBL7700818 0.86 PARP1 (0.36) PARP1NPC1RAB9AKMT2ATP53
SCHEMBL7383364 0.86 NOTUM (0.37) PARP1NPC1RAB9AKMT2ATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6346527-B1 1-BENZOXEPIN DERIVATIVES USED IN THE PREVENTION OF SODIUM AND HYDROGEN ION EXCHANGE; CARDIOVASCULAR, KIDNEY AND BRAIN DISORDER TREATMENT; ARTERIOSCLEROSIS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2002-02-12 US claimed
EP-1073650-A1 GUANIDINE DERIVATIVES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-02-07 EP claimed
WO-1999055690-A1 GUANIDINE DERIVATIVES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1999-11-04 WO claimed