SCHEMBL7702986

SCHEMBL7702986

N=C(N)NC(=O)c1cccc2c1OCCC(C(=O)N=C(N)N)=C2

nearest known ligand 0.38

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.38
SSTR4 P31391 3/20 0.32
HTR2B P41595 2/20 0.31
HTR7 P34969 1/20 0.31
NPC1 O15118 1/20 0.31
RAB9A P51151 1/20 0.31
KMT2A Q03164 1/20 0.31
SLC9A1 P19634 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7697560 0.99 PARP1 (0.37) PARP1SSTR4HTR2BHTR7NPC1
SCHEMBL7702982 0.89 PARP1 (0.43) PARP1SSTR4NPC1RAB9AKMT2A
Hydrochloric Acid SCHEMBL7697554 0.88 PARP1 (0.42) PARP1SSTR4NPC1RAB9AKMT2A
SCHEMBL7701182 0.84 PARP1 (0.43) PARP1HTR2BHTR7SLC9A1
Hydrochloric Acid SCHEMBL7702267 0.82 PARP1 (0.36) PARP1HTR2BHTR7NPC1KMT2A
SCHEMBL7701178 0.82 PARP1 (0.41) PARP1NPC1RAB9AKMT2A
Hydrochloric Acid SCHEMBL7702869 0.81 KDM4E (0.33) PARP1
Hydrochloric Acid SCHEMBL7696598 0.79 RAD52 (0.38) PARP1
SCHEMBL7697131 0.78 PARP1 (0.46) PARP1NPC1RAB9AKMT2A
Hydrochloric Acid SCHEMBL7702260 0.78 PARP1 (0.36) PARP1NPC1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6346527-B1 1-BENZOXEPIN DERIVATIVES USED IN THE PREVENTION OF SODIUM AND HYDROGEN ION EXCHANGE; CARDIOVASCULAR, KIDNEY AND BRAIN DISORDER TREATMENT; ARTERIOSCLEROSIS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2002-02-12 US claimed
EP-1073650-A1 GUANIDINE DERIVATIVES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-02-07 EP claimed
WO-1999055690-A1 GUANIDINE DERIVATIVES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1999-11-04 WO claimed