Atorvastatin

Atorvastatin

SCHEMBL7703363

CC(C)c1c(C(=O)Nc2ccccc2)c(-c2ccccc2)c(-c2ccc(F)cc2)n1CCC(O)CC(O)CC(=O)[O-].CC(C)c1c(C(=O)Nc2ccccc2)c(-c2ccccc2)c(-c2ccc(F)cc2)n1CCC(O)CC(O)CC(=O)[O-].[Ca+2]

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

HMGCR

The experimentally established mechanism targets of Atorvastatin. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HMGCR known ✓ P04035 3/20 0.86
ABCB11 O95342 3/20 1.00
SLCO1B1 Q9Y6L6 3/20 1.00
ABCC3 O15438 2/20 1.00
ABCC4 O15439 2/20 1.00
SLCO1B3 Q9NPD5 2/20 1.00
HDAC1 Q13547 2/20 0.86
HDAC2 Q92769 2/20 0.86
HDAC6 Q9UBN7 2/20 0.86
NR1I2 O75469 1/20 0.86
RHOC P08134 1/20 0.86
CYP3A4 P08684 1/20 0.86
THRB P10828 1/20 0.86
NR1H4 Q96RI1 1/20 0.86
ABCG2 Q9UNQ0 1/20 0.86
PDE6D O43924 3/20 0.74

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Atorvastatin SCHEMBL7037659 1.00 ABCB11 (1.00) ABCB11SLCO1B1ABCC3ABCC4SLCO1B3
Atorvastatin SCHEMBL3832 1.00 ABCB11 (1.00) ABCB11SLCO1B1ABCC3ABCC4SLCO1B3
Atorvastatin SCHEMBL6064039 1.00 ABCB11 (1.00) ABCB11SLCO1B1ABCC3ABCC4SLCO1B3
Atorvastatin SCHEMBL5072672 1.00 ABCB11 (1.00) ABCB11SLCO1B1ABCC3ABCC4SLCO1B3
Atorvastatin SCHEMBL7102147 0.99 ABCB11 (0.98) ABCB11SLCO1B1ABCC3ABCC4SLCO1B3
Atorvastatin SCHEMBL5077129 0.99 ABCB11 (0.98) ABCB11SLCO1B1ABCC3ABCC4SLCO1B3
Atorvastatin SCHEMBL4668716 0.99 ABCB11 (0.98) ABCB11SLCO1B1ABCC3ABCC4SLCO1B3
Atorvastatin SCHEMBL153886 0.99 ABCB11 (0.98) ABCB11SLCO1B1ABCC3ABCC4SLCO1B3
Atorvastatin SCHEMBL1535888 0.99 ABCB11 (0.98) ABCB11SLCO1B1ABCC3ABCC4SLCO1B3
Atorvastatin SCHEMBL28456 0.99 ABCB11 (0.98) ABCB11SLCO1B1ABCC3ABCC4SLCO1B3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002083637-A1 PROCESS FOR THE PRODUCTION OF AMORPHOUS ATORVASTATIN CALCIUM CADILA HEALTHCARE LIMITED (IN) 2002-10-24 WO disclosed