SCHEMBL7703949

SCHEMBL7703949

Cc1cc2c(cc1C(C)(C)Br)C(C)(C)CC(=O)N2

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
RARB P10826 1/20 0.39
RARG P13631 1/20 0.39
HDAC3 O15379 4/20 0.35
HDAC4 P56524 4/20 0.35
HDAC1 Q13547 4/20 0.35
HDAC2 Q92769 4/20 0.35
HDAC8 Q9BY41 4/20 0.35
HDAC6 Q9UBN7 4/20 0.35
HDAC9 Q9UKV0 4/20 0.35
RXRA P19793 1/20 0.32
CMA1 P23946 1/20 0.32
AHR P35869 1/20 0.32
HPGD P15428 1/20 0.30
MAPK1 P28482 1/20 0.30
HSD17B10 Q99714 1/20 0.30
GRIA1 P42261 1/20 0.30
CACNG8 Q8WXS5 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8700087 0.80 BCHE (0.44) RARBRARGHDAC3HDAC4HDAC1
SCHEMBL2242248 0.76 BCHE (0.44) RARBRARGHDAC3HDAC4HDAC1
SCHEMBL12428929 0.76 RARB (0.41) RARBRARGHDAC3HDAC4HDAC1
SCHEMBL26443454 0.76 RARB (0.39) RARBRARGHDAC3HDAC4HDAC1
SCHEMBL7703904 0.74 RARB (0.48) RARBRARGHDAC3HDAC4HDAC1
SCHEMBL9379048 0.70 RARB (0.43) RARBRARGHDAC3HDAC4HDAC1
SCHEMBL11988473 0.69 RARB (0.52) RARBRARGHDAC3HDAC4HDAC1
SCHEMBL2242664 0.69 CYP1A2 (0.49) RARBRARGHDAC3HDAC4HDAC1
SCHEMBL14827606 0.69 HDAC3 (0.44) RARBRARGHDAC3HDAC4HDAC1
SCHEMBL31714583 0.69 RARB (0.40) RARBRARGHDAC3HDAC4HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1228042-A2 TETRAHYDROQUINOLINE DERIVATIVES HAVING RETINOID-LIKE BIOLOGICAL ACTIVITY Allergan Sales, Inc. (US) 2002-08-07 EP disclosed
WO-2001012606-A2 TETRAHYDROQUINOLINE DERIVATIVES HAVING RETINOID-LIKE BIOLOGICAL ACTIVITY ALLERGAN SALES, INC. (US) 2001-02-22 WO disclosed