SCHEMBL7704724

SCHEMBL7704724

CC(C)C(=O)Nc1ccc(-c2n[nH]c3c2Cc2ccccc2-3)cc1

nearest known ligand 0.60

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 9/20 0.60
KDR P35968 3/20 0.60
CDK2 P24941 2/20 0.56
CDK1 P06493 1/20 0.56
NPC1 O15118 2/20 0.47
PDGFRB P09619 2/20 0.44
HIF1A Q16665 1/20 0.44
CCNE2 O96020 1/20 0.44
CDK4 P11802 1/20 0.44
CCND1 P24385 1/20 0.44
CCNE1 P24864 1/20 0.44
POLB P06746 1/20 0.44
RAB9A P51151 1/20 0.44
ALDH1A1 P00352 1/20 0.43
GAA P10253 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7698302 0.89 CHEK1 (0.56) CHEK1KDRCDK2CDK1NPC1
SCHEMBL7697800 0.88 CHEK1 (0.57) CHEK1KDRCDK2CDK1NPC1
SCHEMBL7701864 0.88 CHEK1 (0.54) CHEK1KDRCDK2CDK1NPC1
SCHEMBL7000769 0.87 CHEK1 (0.64) CHEK1KDRCDK2CDK1NPC1
SCHEMBL7092402 0.87 KMT2A (0.55) CHEK1KDRCDK2CDK1PDGFRB
Hydrochloric Acid SCHEMBL7089690 0.86 CHEK1 (0.62) CHEK1KDRCDK2CDK1NPC1
SCHEMBL7705309 0.86 KDR (0.69) CHEK1KDRCDK2CDK1NPC1
SCHEMBL7701530 0.86 CHEK1 (0.57) CHEK1KDRCDK2CDK1NPC1
SCHEMBL7702752 0.85 CHEK1 (0.64) CHEK1KDRCDK2CDK1NPC1
SCHEMBL7705656 0.84 CHEK1 (0.60) CHEK1KDRCDK2CDK1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6462036-B1 INHIBITING SIGNAL TRANSDUCTION BY MODULATING ACTIVITY OF RECEPTOR AND NONRECEPTOR TYROSINE AND SERINE/THREONINE KINASES TO REGULATE AND MODULATE ABNORMAL OR INAPPROPRIATE CELL PROLIFERATION, DIFFERENTIATION, OR METABOLISM BASF AKTIENGESELLSCHAFT (DE) 2002-10-08 US disclosed