SCHEMBL7705017

SCHEMBL7705017

CC1Oc2ccc(C(NC(=O)OC(C)(C)C)C3CCc4ccccc43)cc2N=C1N

nearest known ligand 0.34

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.34
KDM4E B2RXH2 2/20 0.34
RCE1 Q9Y256 1/20 0.34
PLA2G1B P04054 1/20 0.33
MAPT P10636 1/20 0.33
HPGD P15428 1/20 0.33
XBP1 P17861 1/20 0.33
HTT P42858 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
ATG4B Q9Y4P1 1/20 0.33
AAK1 Q2M2I8 3/20 0.32
DRD2 P14416 3/20 0.32
SCN9A Q15858 3/20 0.32
IDO1 P14902 1/20 0.31
ADORA2A P29274 1/20 0.30
SLC8A1 P32418 1/20 0.30
EDNRA P25101 1/20 0.30
BACE1 P56817 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7704833 0.86 KDM4E (0.37) ALDH1A1KDM4ERCE1PLA2G1BMAPT
SCHEMBL7093745 0.80 KDM4E (0.34) ALDH1A1KDM4ERCE1PLA2G1BMAPT
Hydrochloric Acid SCHEMBL6996294 0.78 IDO1 (0.33) IDO1
SCHEMBL7708204 0.76 IDO1 (0.39) ALDH1A1KDM4ERCE1IDO1
SCHEMBL7704912 0.76 ALDH1A1 (0.45) ALDH1A1MAPTHPGDXBP1HTT
SCHEMBL7094224 0.76 ALDH1A1 (0.34) ALDH1A1KDM4ERCE1PLA2G1BMAPT
SCHEMBL7711115 0.75 AAK1 (0.40) ALDH1A1KDM4ERCE1PLA2G1BMAPT
SCHEMBL7704928 0.74 SMYD3 (0.35) IDO1
SCHEMBL7704992 0.73 ALDH1A1 (0.35) ALDH1A1KDM4ERCE1PLA2G1BMAPT
SCHEMBL7091668 0.73 IDO1 (0.34) ALDH1A1KDM4EIDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6365736-B1 TREATMENT OF NERVOUS SYSTEM DISORDERS, CARDIOVASCULAR DISORDERS AND FOR ACTIVITY AS NO-SYNTHASES (NOS) INHIBITORS. SCHERING AKTIENGESELLSCHAFT (DE) 2002-04-02 US disclosed