SCHEMBL7706963

SCHEMBL7706963

CC(C)(C)OC(=O)[C@H](Cc1ccc(CCCCCC(=O)NC2=CCCCN2)s1)NC(=O)OCc1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 3/20 0.44
ITGAV P06756 3/20 0.44
ITGA2B P08514 1/20 0.44
SYK P43405 1/20 0.36
KLK7 P49862 3/20 0.36
HDAC1 Q13547 4/20 0.35
KLK5 Q9Y337 2/20 0.35
CTSL P07711 2/20 0.35
CTSB P07858 1/20 0.35
CTSS P25774 1/20 0.35
HDAC3 O15379 1/20 0.35
HDAC4 P56524 1/20 0.35
HDAC7 Q8WUI4 1/20 0.35
HDAC2 Q92769 1/20 0.35
HDAC10 Q969S8 1/20 0.35
HDAC11 Q96DB2 1/20 0.35
HDAC8 Q9BY41 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35
HDAC9 Q9UKV0 1/20 0.35
HDAC5 Q9UQL6 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7706968 1.00 ITGB3 (0.44) ITGB3ITGAVITGA2BSYKKLK7
SCHEMBL5561128 0.86 ITGB3 (0.60) ITGB3ITGAVITGA2B
SCHEMBL5567560 0.85 ITGB3 (0.61) ITGB3ITGAVITGA2B
SCHEMBL5566427 0.83 SYK (0.45) ITGB3ITGAVITGA2BSYKCTSL
SCHEMBL5566516 0.82 SYK (0.45) ITGB3ITGAVITGA2BSYKCTSL
SCHEMBL5567726 0.77 ITGB3 (0.69) ITGB3ITGAVITGA2B
SCHEMBL14546828 0.77 ITGB3 (0.69) ITGB3ITGAVITGA2B
SCHEMBL5561642 0.76 ITGB3 (0.70) ITGB3ITGAVITGA2B
SCHEMBL5562060 0.74 ITGB3 (0.53) ITGB3ITGAVITGA2B
SCHEMBL5562064 0.74 ITGB3 (0.53) ITGB3ITGAVITGA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1240161-A1 THIENYLALANINE DERIVATIVES AS INHIBITORS OF CELL ADHESION Aventis Pharma Deutschland GmbH (DE) 2002-09-18 EP disclosed
WO-2001044237-A1 THIENYLALANINE DERIVATIVES AS INHIBITORS OF CELL ADHESION AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2001-06-21 WO disclosed