SCHEMBL7707683

SCHEMBL7707683

O=C(O)CN1CCN(CCc2ccccc2OCc2cc(C(F)(F)F)cc(C(F)(F)F)c2)CC1

nearest known ligand 0.55

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 16/20 0.55
KCNH2 Q12809 2/20 0.47
SLC1A5 Q15758 1/20 0.43
FPR2 P25090 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7705623 0.92 TACR1 (0.56) TACR1KCNH2SLC1A5
SCHEMBL7705390 0.89 TACR1 (0.60) TACR1KCNH2SLC1A5
SCHEMBL7705827 0.89 TACR1 (0.56) TACR1KCNH2
SCHEMBL7699781 0.88 TACR1 (0.61) TACR1KCNH2FPR2
SCHEMBL7699901 0.88 TACR1 (0.59) TACR1KCNH2SLC1A5
SCHEMBL7704886 0.87 TACR1 (0.48) TACR1
SCHEMBL7699833 0.87 TACR1 (0.49) TACR1KCNH2SLC1A5
SCHEMBL7704919 0.84 TACR1 (0.54) TACR1
SCHEMBL7705237 0.84 KCNH2 (0.46) KCNH2
SCHEMBL7699915 0.84 MRGPRX4 (0.51) KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1242399-A1 $g(a)-ARYLETHYLPIPERAZINE DERIVATIVES AS NEUROKININ ANTAGONISTS UCB S.A. (BE) 2002-09-25 EP disclosed
WO-2001046167-A1 α-ARYLETHYLPIPERAZINE DERIVATIVES AS NEUROKININ ANTAGONISTS UCB, S.A. (BE) 2001-06-28 WO disclosed