SCHEMBL7705237

SCHEMBL7705237

O=C(O)CN1CCN(CCc2ccccc2OCc2cc(Br)cc(Br)c2)CC1

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 5/20 0.46
SIGMAR1 Q99720 3/20 0.44
CFD P00746 1/20 0.43
F11 P03951 1/20 0.43
TPSB2 P20231 1/20 0.43
ALDH1A1 P00352 1/20 0.42
PTPN2 P17706 1/20 0.42
PTPN1 P18031 1/20 0.42
HTR1A P08908 1/20 0.40
DRD2 P14416 1/20 0.40
PTGER1 P34995 1/20 0.40
PTGER4 P35408 1/20 0.40
PTGER3 P43115 1/20 0.40
PTGER2 P43116 1/20 0.40
HRH3 Q9Y5N1 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.39
HRH1 P35367 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7707683 0.84 TACR1 (0.55) KCNH2
SCHEMBL16396757 0.77 CFD (0.62) CFDF11TPSB2PTGER1PTGER4
SCHEMBL7705623 0.75 TACR1 (0.56) KCNH2
SCHEMBL7705827 0.73 TACR1 (0.56) KCNH2SIGMAR1
SCHEMBL7705390 0.73 TACR1 (0.60) KCNH2SIGMAR1
SCHEMBL7699781 0.72 TACR1 (0.61) KCNH2ALDH1A1PTPN2PTPN1
SCHEMBL7699901 0.72 TACR1 (0.59) KCNH2SIGMAR1
SCHEMBL16396440 0.71 CFD (0.59) CFDF11TPSB2PTGER1PTGER4
SCHEMBL16397056 0.71 CFD (0.49) CFDF11TPSB2ALDH1A1PTGER1
SCHEMBL7704886 0.71 TACR1 (0.48) PTGER1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1242399-A1 $g(a)-ARYLETHYLPIPERAZINE DERIVATIVES AS NEUROKININ ANTAGONISTS UCB S.A. (BE) 2002-09-25 EP claimed
WO-2001046167-A1 α-ARYLETHYLPIPERAZINE DERIVATIVES AS NEUROKININ ANTAGONISTS UCB, S.A. (BE) 2001-06-28 WO claimed